BDBM50016958 1-(4-Fluoro-phenyl)-4-(4-thieno[3,2-c]pyridin-4-yl-piperazin-1-yl)-butan-1-ol::CHEMBL15560

SMILES OC(CCCN1CCN(CC1)c1nccc2sccc12)c1ccc(F)cc1

InChI Key InChIKey=YZSXHWKLZRAMBW-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50016958   

Target5-hydroxytryptamine receptor 1A/1B/1D/1F(Rat)
Bristol-Myers

Curated by ChEMBL
LigandPNGBDBM50016958(CHEMBL15560 | 1-(4-Fluoro-phenyl)-4-(4-thieno[3,2-...)
Affinity DataIC50: 3.80nMAssay Description:Ability to bind at 5-hydroxytryptamine 1 receptor of rat hippocampus by displacing [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandPNGBDBM50016958(CHEMBL15560 | 1-(4-Fluoro-phenyl)-4-(4-thieno[3,2-...)
Affinity DataIC50: 23nMAssay Description:Ability to bind at alpha-1 adrenergic receptor by displacing [3H]WB-4101More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandPNGBDBM50016958(CHEMBL15560 | 1-(4-Fluoro-phenyl)-4-(4-thieno[3,2-...)
Affinity DataIC50: 5.80nMAssay Description:Ability to bind at serotonin 5-hydroxytryptamine 2 receptors of rat hippocampus by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Bristol-Myers

Curated by ChEMBL
LigandPNGBDBM50016958(CHEMBL15560 | 1-(4-Fluoro-phenyl)-4-(4-thieno[3,2-...)
Affinity DataIC50: 72nMAssay Description:Ability to bind at dopamine receptor D2 of rat corpus striatum by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed