BDBM50006255 CHEMBL418353

SMILES CCCCC\C=C/C\C=C/C\C=C/C\C=C/CCCC(=O)NC1CC1

InChI Key InChIKey=GLGAUBPACOBAMV-UHFFFAOYSA-N

Data  4 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50006255   

TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50006255(CHEMBL418353)
Affinity DataEC50:  398nMAssay Description:Displacement of [35S]GTP-gamma-S from rat cerebellar CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50006255(CHEMBL418353)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]-CP55940 from CB1 receptor of rat cerebellar membranes by liquid scintillation counting in presence of serine protease inhibitor ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Kuopio

Curated by ChEMBL
LigandPNGBDBM50006255(CHEMBL418353)
Affinity DataKi:  2.70nMAssay Description:Binding affinity towards rat brain cannabinoid receptor 1 in the presence of PMSF upon incubation for 15 min at 4 degree C in pH 7.4 using [3H]CP-559...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Mouse)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50006255(CHEMBL418353)
Affinity DataKi:  157nMAssay Description:Binding affinity towards mouse spleen cannabinoid receptor 2 in the presence of PMSF upon incubation for 15 min at 4 degree C in pH 7.4 using [3H]CP-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50006255(CHEMBL418353)
Affinity DataKi:  715nMAssay Description:Displacement of [3H]-CP55940 from CB2 receptor of rat spleen membranes by liquid scintillation counting in presence of serine protease inhibitor PMSFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed