BDBM492927 US10981898, Example 20

SMILES CC(C)[Si](C#Cc1ccc(CN2C(=O)c3cc(ccc3C2(OCC2(CO)CC2)c2ccc(Cl)cc2)C(C)(C)O)cc1)(C(C)C)C(C)C

InChI Key InChIKey=MSTKICFKUWVYLG-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 492927   

TargetCellular tumor antigen p53 [1-83]/E3 ubiquitin-protein ligase Mdm2 [1-188](Human)
Astex Therapeutics

US Patent

LigandBDBM492927(US10981898, Example 20)Copy SMILESCopy InChI

Affinity DataIC50: 11nMAssay Description:The ELISA assay was performed in streptavidin coated plates which were preincubated with 200 μl per well of 1 μg ml−1 biotinylated IP...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
10/26/2021
Entry Details
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