BDBM469657 N-tert-Butyl-4-[[2-(2-hydroxyphenyl)acetyl]amino]pyridine-2-carboxamide::US11364246, Example 1::US20200361871A1, Example 1

SMILES CC(C)(C)NC(=O)c1cc(NC(=O)Cc2ccccc2O)ccn1

InChI Key InChIKey=MEKPLZGVNVGOOQ-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 469657   

TargetAnoctamin-1(Human)
Enterprise Therapeutics

US Patent
LigandPNGBDBM469657(US20200361871A1, Example 1 | N-tert-Butyl-4-[[2-(2...)
Affinity DataEC50:  210nMAssay Description:Compound activity was quantified by measuring the increase in current upon compound addition and expressing this as a percentage increase of baseline...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAnoctamin-1(Human)
Enterprise Therapeutics

US Patent
LigandPNGBDBM469657(US20200361871A1, Example 1 | N-tert-Butyl-4-[[2-(2...)
Affinity DataEC50:  210nMAssay Description:Cell Culture and PreparationFisher rat thyroid (FRT) cells stably expressing human TMEM16A (TMEM16Aabc variant; Dr Luis Galietta, Insituto Giannina, ...More data for this Ligand-Target Pair
In DepthDetails
US Patent