BDBM458507 2-(2-Fluoro-6-methoxyphenyl)-N-(1-methyl-4-(2-((methylamino)methyl)phenyl)-1H-indazol-5-yl)pyrimidine-4-carboxamide::US10745388, Example 15

SMILES CNCc1ccccc1-c1c(NC(=O)c2ccnc(n2)-c2c(F)cccc2OC)ccc2n(C)ncc12

InChI Key InChIKey=NIXHGNOEARVEHJ-UHFFFAOYSA-N

Data  1 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 458507   

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Incyte

US Patent

LigandBDBM458507(2-(2-Fluoro-6-methoxyphenyl)-N-(1-methyl-4-(2-((me...)Copy SMILESCopy InChI

Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
4/13/2021
Entry Details
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