BDBM457866 1-(1-(2-chlorobenzyl)piperidin-4-yl)-3-(cyclopropylmethyl)-5-methyl-1H-benzo[d]imidazol-2(3H)-one::US10751335, Example 28
SMILES Cc1ccc2n(C3CCN(Cc4ccccc4Cl)CC3)c(=O)n(CC3CC3)c2c1
InChI Key InChIKey=GCDUWEOWDBFAQN-UHFFFAOYSA-N
Data 2 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 457866
Affinity DataEC50: 558nMAssay Description:A standard [35S]GTPγS binding assay in membranes prepared from CHO cells expressing the human MOR was performed in a concentration response mann...More data for this Ligand-Target Pair
Affinity DataEC50: 253nMAssay Description:he CisBio cAMP cell based assay kit that uses HTRF technology was utilized to assess MOR-mediated inhibition of cAMP. Assays were performed according...More data for this Ligand-Target Pair