BDBM445542 2-{8-Fluoro-5-[(5-methyl-1,2-oxazol-3-yl)(oxan-4-yl)methyl]-7-[4-(2H3)methyl-1-methyl-1H-1,2,3-triazol-5-yl]-5H-pyrido[3,2-b]indol-3-yl}propan-2-ol::US10683290, Example 34::US10683290, Example 35
SMILES Cc1cc(no1)C(C1CCOCC1)n1c2cc(-c3c(C)nnn3C)c(F)cc2c2ncc(cc12)C(C)(C)O
InChI Key InChIKey=OPGYUCHNVCWIIN-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 445542
Affinity DataIC50: 1nMAssay Description:All assay components were dissolved in buffer composition 20 mM Hepes pH 7.5, 150 mM NaCl, 5 mM DTT, 0.005% Tween 20, and 100 ug/ml BSA for BRD4 (1-4...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:All assay components were dissolved in buffer composition 20 mM Hepes pH 7.5, 150 mM NaCl, 5 mM DTT, 0.005% Tween 20, and 100 ug/ml BSA for BRD4 (1-4...More data for this Ligand-Target Pair