BDBM436031 5-[2-Methyl-3-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]-1,3-::US10611730, Example 203

SMILES Cc1noc(n1)-c1cccc(-c2ccc3[nH]c(=O)[nH]c3c2)c1C

InChI Key InChIKey=AFXKJXJXEXUZKY-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 436031   

TargetVoltage-dependent calcium channel gamma-8 subunit(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM436031(US10611730, Example 203 | 5-[2-Methyl-3-(3-methyl-...)
Affinity DataIC50: 39.8nMAssay Description:This assay was used to test compounds for their ability to inhibit TARP γ8 dependent AMPA receptor activity. The AMPA receptor is a non-selectiv...More data for this Ligand-Target Pair
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Date in BDB:
12/7/2020
Entry Details
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