BDBM436029 5-(3-(3-Cyclopropyl-1,2,4-oxadiazol-5-yl)-2-methylphenyl)-1H-::US10611730, Example 201

SMILES Cc1c(cccc1-c1ccc2[nH]c(=O)[nH]c2c1)-c1nc(no1)C1CC1

InChI Key InChIKey=OILJIMBLIDBMKG-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 436029   

TargetVoltage-dependent calcium channel gamma-8 subunit(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM436029(US10611730, Example 201 | 5-(3-(3-Cyclopropyl-1,2,...)
Affinity DataIC50: 10nMAssay Description:This assay was used to test compounds for their ability to inhibit TARP γ8 dependent AMPA receptor activity. The AMPA receptor is a non-selectiv...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2020
Entry Details
Go to US Patent