BDBM434075 US10562890, Compound Al-14-95

SMILES FC(F)(F)Oc1ccc2[nH]c(nc2c1)-c1ccc(OCCN2CCN(Cc3ccccc3)CC2)cn1

InChI Key InChIKey=HUTFNFMGRNFVCG-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 434075   

TargetRunt-related transcription factor 1(Human)
University of Virginia Patent Foundation

US Patent
LigandPNGBDBM434075(US10562890, Compound Al-14-95)
Affinity DataIC50: 2.65E+3nMAssay Description:FRET assay can be used to effectively monitor the inhibition of CBF binding to the Runt domain of RUNX proteins (as well as for CBFβ-SMMHC bindi...More data for this Ligand-Target Pair
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Date in BDB:
11/22/2020
Entry Details
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