BDBM406388 N-(tert-Butylsulfonyl)-2-((rac-trans)-4-hydroxy-3-(thiazol-4-ylmethyl)chroman-7-yl)benzamide::US10336733, Example 32::US10336733, Example 34

SMILES CC(C)(C)S(=O)(=O)NC(=O)c1ccccc1-c1ccc2[C@H](O)[C@@H](Cc3cscn3)COc2c1

InChI Key InChIKey=PGVLVBJRARVNRB-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 406388   

TargetLeukotriene B4 receptor 1(Human)
Merk Sharp & Dohme

US Patent
LigandPNGBDBM406388(US10336733, Example 34 | N-(tert-Butylsulfonyl)-2-...)
Affinity DataEC50:  11nMAssay Description:The ability of compounds to antagonize the human BLT1 receptor was determined using a kit to measure changes in intracellular cyclic AMP levels (cAMP...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetLeukotriene B4 receptor 1(Human)
Merk Sharp & Dohme

US Patent
LigandPNGBDBM406388(US10336733, Example 34 | N-(tert-Butylsulfonyl)-2-...)
Affinity DataEC50:  9nMAssay Description:The ability of compounds to antagonize the human BLT1 receptor was determined using a kit to measure changes in intracellular cyclic AMP levels (cAMP...More data for this Ligand-Target Pair
In DepthDetails
US Patent