BDBM406365 4-Fluoro-2-((3S,4R or 3R,4S)-4-hydroxy-3-(pyridin-2-ylmethyl)chroman-7-yl)-N-((1-methylcyclopropyl)sulfonyl)benzamide::US10336733, Example 9

SMILES CC1(CC1)S(=O)(=O)NC(=O)c1ccc(F)cc1-c1ccc2[C@H](O)[C@@H](Cc3ccccn3)COc2c1

InChI Key InChIKey=PLHBWJXLGZYYHG-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 406365   

TargetLeukotriene B4 receptor 1(Human)
Merk Sharp & Dohme

US Patent
LigandPNGBDBM406365(4-Fluoro-2-((3S,4R or 3R,4S)-4-hydroxy-3-(pyridin-...)
Affinity DataEC50:  4nMAssay Description:The ability of compounds to antagonize the human BLT1 receptor was determined using a kit to measure changes in intracellular cyclic AMP levels (cAMP...More data for this Ligand-Target Pair
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US Patent