BDBM396722 6-(6'-methyl-[2,2'-bipyridin]-3- yl)imidazo[1,2-a]pyridine-3-carboxylic acid::US9981944, Example 67

SMILES Cc1cccc(n1)-c1ncccc1-c1ccc2ncc(C(O)=O)n2c1

InChI Key InChIKey=QQFLQHVUKANAAG-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 396722   

TargetTGF-beta receptor type-1 [T204D](Human)
Rigel Pharmaceuticals

US Patent
LigandPNGBDBM396722(US9981944, Example 67 | 6-(6'-methyl-[2,2'-bipyrid...)
Affinity DataIC50: 4nMAssay Description:Assays for the compounds reported below were conducted in 1536-well plates and 2 mL reactions are prepared from addition of HIS-TGFβR1 T204D or ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent