BDBM359715 N-(4-(2,6-dimethoxyphenyl)-5-(6-methoxy-2-pyridinyl)-4H-1,2,4-triazol-3-::US10221162, Example 4.02

SMILES COc1cccc(n1)C(=O)NN\C(NS(C)(=O)=O)=N\c1c(OC)cccc1OC

InChI Key InChIKey=BEDGLBITLAXPQN-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 359715   

TargetApelin receptor(Human)
Amgen

US Patent
LigandPNGBDBM359715(N-(4-(2,6-dimethoxyphenyl)-5-(6-methoxy-2-pyridiny...)
Affinity DataEC50:  220nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV -3 expression vector (Si...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
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