BDBM352390 5-[5-(7-Ethyl-7H-imidazo[4,5-c]pyridazin-4-yl)-2-fluorophenyl]-6-methoxy-2-methyl-2,3-dihydro-1H-isoindol-1-one::US9802945, 1

SMILES CCn1cnc2c(cnnc12)-c1ccc(F)c(c1)-c1cc2CN(C)C(=O)c2cc1CO

InChI Key InChIKey=ZXBDRFOZYPKXKS-UHFFFAOYSA-N

Data  1 KI

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 352390   

TargetGamma-aminobutyric acid receptor subunit alpha-2(Human)
Pfizer

US Patent

LigandBDBM352390(5-[5-(7-Ethyl-7H-imidazo[4,5-c]pyridazin-4-yl)-2-f...)Copy SMILESCopy InChI

Affinity DataKi:  6.60nMAssay Description:The affinity of the test compounds was determined by radioligand competition binding assay, using the known compound [3H]Ro-15-1788 (Flumazenil) (Per...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
10/1/2019
Entry Details
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