BDBM308048 5-(4-butoxyphenyl)-1-(H- imidazo[1,2-a]pyridin-7- yl)imidazolidin-2-one::US9650362, 55

SMILES CCCCOc1ccc(cc1)C1CNC(=O)N1c1ccn2ccnc2c1

InChI Key InChIKey=DOMIMUPMZJUIBB-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 308048   

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandPNGBDBM308048(US9650362, 55 | 5-(4-butoxyphenyl)-1-(H- imidazo[1...)
Affinity DataIC50: 397nMAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometrical...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Probiodrug

US Patent
LigandPNGBDBM308048(US9650362, 55 | 5-(4-butoxyphenyl)-1-(H- imidazo[1...)
Affinity DataKi:  75nMAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometrical...More data for this Ligand-Target Pair
In DepthDetails
US Patent