BDBM30066 triazolothiadiazine, 6G

SMILES COc1ccc(cc1OC)-c1nnc2SCC(=Nn12)c1ccccc1OC

InChI Key InChIKey=FRYZTSQSRVHSPO-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 30066   

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
Nih

LigandBDBM30066(triazolothiadiazine, 6G)Copy SMILESCopy InChI

Affinity DataIC50: 8.90E+3nMpH: 7.2 T: 2°CAssay Description:Inhibition of PDE4A was performed using IMAP technology (Molecular Devices, CA). PDE4A1A mixture was dispensed into 1536-well black/solid bottom assa...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
7/4/2009
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