BDBM297842 (−)-trans-7-(2-Methylpiperidin-4-yl)-5-oxo-4,5-dihydropyrazolo[1,5-a]pyrimidine-3-carbonitrile trifluoroacetate::US10118930, Example 65

SMILES CC1CC(CCN1)c1cc(=O)[nH]c2c(cnn12)C#N

InChI Key InChIKey=RVXFYHDUCASLKN-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 297842   

TargetTissue-type plasminogen activator(Human)
Bayer Pharma Aktiengesellschaft

US Patent
LigandPNGBDBM297842(US10118930, Example 65 | (−)-trans-7-(2-Meth...)
Affinity DataIC50: 12nMAssay Description:The clot-lysis test system configures the kinetics of clot formation and degradation in vitro and allows quantifying modulation of the process by sel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
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