BDBM289929 3-[1-(2-{6-[5-(2H-Pyrazol-3-yl)- pyridin-2-yloxy]-2,3-dihydro- benzofuran-3-yl}-ethyl)-piperidin- 4-yl]-oxazolidin-2-one::US9573957, Example 69

SMILES O=C1OCCN1C1CCN(CCC2COc3cc(Oc4ccc(cn4)-c4ccn[nH]4)ccc23)CC1

InChI Key InChIKey=MBJLUUJSGCMGEZ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 289929   

TargetLeukotriene A-4 hydrolase(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM289929(3-[1-(2-{6-[5-(2H-Pyrazol-3-yl)- pyridin-2-yloxy]-...)
Affinity DataIC50: 0.75nMpH: 7.5 T: 2°CAssay Description:The compounds of the invention are assessed for the ability to interact with human LTA4 hydrolase in an enzymatic assay that measures the ability of ...More data for this Ligand-Target Pair
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US Patent