BDBM289507 5-(2-(cyclopropyl- methyl)-1-(3-(4- methylpiperazin-1-yl)- bicyclo[1.1.1]pentan-1- yl)-1H-imidazol-4-yl)- 3-(trifluoromethoxy)- pyridin-2-amine::US10093664, Example 72

SMILES CN1CCN(CC1)C12CC(C1)(C2)n1cc(nc1CC1CC1)-c1cnc(N)c(OC(F)(F)F)c1

InChI Key InChIKey=DTYHKSLSXPMHOR-UHFFFAOYSA-N

Data  1 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 289507   

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandPNGBDBM289507(US10093664, Example 72 | 5-(2-(cyclopropyl- methyl...)
Affinity DataKd:  19nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
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