BDBM289470 3-(difluoromethoxy)-5- (2-isobutyl-1-(3- morpholinobicyclo- [1.1.1]pentan-1-yl)-1H- imidazol-4-yl)pyridin- 2-amine::US10093664, Example 46

SMILES CC(C)Cc1nc(cn1C12CC(C1)(C2)N1CCOCC1)-c1cnc(N)c(OC(F)F)c1

InChI Key InChIKey=SJEIJBOBGUGBEZ-UHFFFAOYSA-N

Data  1 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 289470   

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandPNGBDBM289470(US10093664, Example 46 | 3-(difluoromethoxy)-5- (2...)
Affinity DataKd:  29nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
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