BDBM289431 5-(2-cyclopropyl-1-(3-(4-methylpiperazin-1-yl)bicyclo[1.1.1]pentan-1-yl)-1H-imidazol-4-yl)-3-(trifluoromethoxy)pyridin-2-amine::US10093664, Example 12

SMILES CN1CCN(CC1)C12CC(C1)(C2)n1cc(nc1C1CC1)-c1cnc(N)c(OC(F)(F)F)c1

InChI Key InChIKey=FPTBZVDMXLZGSQ-UHFFFAOYSA-N

Data  1 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 289431   

TargetMitogen-activated protein kinase kinase kinase 12(Human)
The University of Texas System

US Patent
LigandPNGBDBM289431(US10093664, Example 12 | 5-(2-cyclopropyl-1-(3-(4-...)
Affinity DataKd:  20nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
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