BDBM278438 (2S)-2-methoxy-2-(4- methoxyphenyl)-N-[5-[[(3R)- 1-(1,2,4-triazin-3- yl)pyrrolidin-3-yl]amino]- 1,3,4-thiadiazol-2- yl]acetamide::US10040788, Example 24::US10294221, Example 24
SMILES CO[C@H](C(=O)Nc1nnc(N[C@@H]2CCN(C2)c2nccnn2)s1)c1ccc(OC)cc1
InChI Key InChIKey=GFVLMJJDMPLIDT-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 278438
Affinity DataIC50: 74.7nMpH: 7.8Assay Description:A Glutamate Oxidase/AmplexRed coupled assay was used to measure the ability of compounds to bind to and inhibit the activity of GLS1 in vitro. 6His t...More data for this Ligand-Target Pair
Affinity DataIC50: 74.7nMAssay Description:A Glutamate Oxidase/AmplexRed coupled assay was used to measure the ability of compounds to bind to and inhibit the activity of GLS1 in vitro. 6His t...More data for this Ligand-Target Pair