BDBM276766 (s)-3-bromo-N-(4-(N-(2-oxotetrahydrofuran-3-yl)sulfamoyl)phenyl)thiophene-2-carboxamide ::US10071994, Compound 10

SMILES Brc1ccsc1C(=O)Nc1ccc(cc1)S(=O)(=O)NC1CCOC1=O

InChI Key InChIKey=XKNGCXNLYGUJCO-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 276766   

TargetSigma-54-dependent Fis family transcriptional regulator(Chromobacterium violaceum)
Institute of Pharmacology and Toxicology Academy of Military Medical Sciences P.L.A. China

US Patent
LigandPNGBDBM276766(US10071994, Compound 10 | (s)-3-bromo-N-(4-(N-(2-o...)
Affinity DataIC50: 1.35E+4nMAssay Description:2.1 The wells of a 12-well plate were marked as initial concentration group, 2, 4, 8, 16, 32, 64, 128, and 256 fold diluted group, DMSO group, and a ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
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