BDBM272934 (S)-1-(1-(2- aminobenzo[d]thiazol- 6-yl)-7,8,9,10- tetrahydro-6-oxa- 2,10a- diazacycloocta[cd]inden- 4-yl)pyrrolidine- 2-carboxamide::US10065970, Compound 239::US10435414, Compound 239

SMILES NC(=O)[C@@H]1CCCN1c1cc2OCCCCn3c(nc(c1)c23)-c1ccc2nc(N)sc2c1

InChI Key InChIKey=CRFQXSJEFRFTEY-UHFFFAOYSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 272934   

LigandPNGBDBM272934((S)-1-(1-(2- aminobenzo[d]thiazol- 6-yl)-7,8,9,10-...)
Affinity DataKi:  0.0350nMAssay Description:PI3K Binding assays are intended for determining the biochemical potency of small molecule PI3K inhibitors. The PI3K lipid kinase reaction is perform...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2018
Entry Details
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LigandPNGBDBM272934((S)-1-(1-(2- aminobenzo[d]thiazol- 6-yl)-7,8,9,10-...)
Affinity DataKi:  0.0350nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details
Go to US Patent