BDBM212714 US9556111, Table 1.12::US9951033, Compound Table 1.15

SMILES OC(=O)c1csc(CN(Cc2cccc(c2)C(F)(F)F)Cc2ccccc2F)n1

InChI Key InChIKey=KIKNZNAERCDRHK-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 212714   

TargetA-kinase anchor protein 7 isoform gamma(Human)
Universitetet I Oslo

US Patent
LigandPNGBDBM212714(US9556111, Table 1.12 | US9951033, Compound Table ...)
Affinity DataEC50:  2.16E+5nMAssay Description:Stable and optimal assay conditions were determined by cross-titrating GST-AKAP18δ and biotinylated PLB using 10 μg/ml glutathione acceptor...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetA-kinase anchor protein 7 isoform gamma(Mouse)
Universitetet I Oslo

US Patent
LigandPNGBDBM212714(US9556111, Table 1.12 | US9951033, Compound Table ...)
Affinity DataEC50:  2.16E+5nMAssay Description:Stable and optimal assay conditions were determined by cross-titrating GST-AKAP18 δ and biotinylated PLB using 10 μg/ml glutathione accepto...More data for this Ligand-Target Pair
In DepthDetails
US Patent