BDBM210899 US9273043, A155(a)

SMILES C[C@H]1CN(CCN1C(=O)Nc1nc2cc(F)ccc2s1)c1ncc(cc1F)[C@H](O)CO

InChI Key InChIKey=GVENNMJXQHKHOV-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 210899   

LigandPNGBDBM210899(US9273043, A155(a))
Affinity DataIC50: 96nMpH: 7.4Assay Description:One day prior to assay, TRPV1/CHO cells were seeded in 96-well clear-bottom black plates (20,000 cells/well) in growth media. On the day of the exper...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2017
Entry Details
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LigandPNGBDBM210899(US9273043, A155(a))
Affinity DataIC50: 700nMT: 2°CAssay Description:Briefly, hTRPV1/CHO cells were cultured in growth media in a tissue culture dish at 37° C. in a CO2 incubator. On the day of the assay, culture m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/30/2017
Entry Details
Go to US Patent