BDBM184915 BDBM50364134::US9156811, DDD87762

SMILES Cc1nn(C)c(C)c1NS(=O)(=O)c1c(Cl)cc(cc1Cl)-c1cccc2CNCCc12

InChI Key

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 184915   

TargetGlycylpeptide N-tetradecanoyltransferase(Trypanosoma brucei brucei (strain 927/4 GUTat10.1))
Univeristy of Dundee

US Patent
LigandPNGBDBM184915(US9156811, DDD87762 | BDBM50364134)
Affinity DataIC50: 2.60E+3nMpH: 7.4 T: 2°CAssay Description:Measurements were performed using a modification of the scintillation proximity assay platform described previously by Georgopapadakou, N. H. et al. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2016
Entry Details
Go to US Patent

TargetGlycylpeptide N-tetradecanoyltransferase 1(Human)
University of Dundee

Curated by ChEMBL
LigandPNGBDBM184915(US9156811, DDD87762 | BDBM50364134)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed