BDBM17593 CHEMBL170733::N'-[(2S,3S)-3-amino-2-hydroxy-4-[(2-methylpropyl)sulfanyl]butanoyl]-3-chlorobenzohydrazide::bestatin-type inhibitor, 8

SMILES CC(C)CSC[C@@H](N)[C@H](O)C(=O)NNC(=O)c1cccc(Cl)c1

InChI Key InChIKey=JUMYLWKXTXAZGY-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 17593   

TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17593(CHEMBL170733 | N'-[(2S,3S)-3-amino-2-hydroxy-4-[(2...)
Affinity DataIC50: 130nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2007
Entry Details
PubMed
TargetMethionine aminopeptidase 1(Human)
Abbott Laboratories

LigandPNGBDBM17593(CHEMBL170733 | N'-[(2S,3S)-3-amino-2-hydroxy-4-[(2...)
Affinity DataIC50: 8.10E+3nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase activity by monitoring the production of free methionine with L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2007
Entry Details
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17593(CHEMBL170733 | N'-[(2S,3S)-3-amino-2-hydroxy-4-[(2...)
Affinity DataIC50: 130nMAssay Description:Inhibitory activity against human methionine aminopeptidase-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMethionine aminopeptidase 1(Human)
Abbott Laboratories

LigandPNGBDBM17593(CHEMBL170733 | N'-[(2S,3S)-3-amino-2-hydroxy-4-[(2...)
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibitory activity against human methionine aminopeptidase-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed