BDBM17467 1,2,3-triazole analogue, 23::5-(3-bromophenyl)-1H-1,2,3-triazole
SMILES Brc1cccc(c1)-c1c[nH]nn1
InChI Key InChIKey=BKJXSQXZIOTRTP-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 17467
TargetIndoleamine 2,3-dioxygenase 1(Mouse)
Ludwig Center For Cancer Research of The University of Lausanne
Curated by ChEMBL
Ludwig Center For Cancer Research of The University of Lausanne
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of mouse IDO1 in P815 clone 6 cells by HPLC analysisMore data for this Ligand-Target Pair
TargetIndoleamine 2,3-dioxygenase 1(Human)
Ludwig Center For Cancer Research of The University of Lausanne
Curated by ChEMBL
Ludwig Center For Cancer Research of The University of Lausanne
Curated by ChEMBL
Affinity DataIC50: 940nMAssay Description:Inhibition of human IDO1 transfected in mouse P815B clone-6 cells by HPLC analysisMore data for this Ligand-Target Pair
TargetTryptophan 2,3-dioxygenase(Mouse)
Ludwig Center For Cancer Research of The University of Lausanne
Curated by ChEMBL
Ludwig Center For Cancer Research of The University of Lausanne
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mouse TDO in P815 clone 12 cells by HPLC analysisMore data for this Ligand-Target Pair
TargetTryptophan 2,3-dioxygenase(Human)
Ludwig Center For Cancer Research of The University of Lausanne
Curated by ChEMBL
Ludwig Center For Cancer Research of The University of Lausanne
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human TDO transfected in mouse P815B clone 19 cells by HPLC analysisMore data for this Ligand-Target Pair
TargetIndoleamine 2,3-dioxygenase 1(Human)
Ludwig Center For Cancer Research of The University of Lausanne
Curated by ChEMBL
Ludwig Center For Cancer Research of The University of Lausanne
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMpH: 6.5Assay Description:Inhibition of human recombinant N-terminal His-tagged IDO1 (Ala2 to Gly403) overexpressed in Escherichia coli BL21 at pH 6.5 after 60 mins by HPLC an...More data for this Ligand-Target Pair
Affinity DataKi: 4nM ΔG°: -11.3kcal/molepH: 7.5 T: 2°CAssay Description:MetAP2 activity was monitored by measuring the initial velocity of turnover of the artificial substrate Met-AMC. Assays were performed in 96-well mi...More data for this Ligand-Target Pair