BDBM150200 US8980905, 108::US9637499, Compound 108

SMILES [O-][n+]1cc(Cl)c(CC(=O)c2ccc(OC(F)F)c3OC4(CCS(=O)(=O)CC4)Oc23)c(Cl)c1

InChI Key InChIKey=ZININGNRPUGNSL-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 150200   

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
Leo Pharma

US Patent
LigandPNGBDBM150200(US8980905, 108 | US9637499, Compound 108)
Affinity DataIC50: 16nMAssay Description:Human recombinant PDE4 (Genbank accession no NM006203) was incubated for 1 hour, with the test compound at concentrations up to 10 μM, with cAMP...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Human)
Leo Pharma

US Patent
LigandPNGBDBM150200(US8980905, 108 | US9637499, Compound 108)
Affinity DataIC50: 16nMAssay Description:Human recombinant PDE4 (Genbank accession no NM_006203) was incubated for 1 hour, with the test compound at concentrations up to 10 μM, with cAM...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Guangdong Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM150200(US8980905, 108 | US9637499, Compound 108)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of PDE3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A [559-660](Human)
Guangdong Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM150200(US8980905, 108 | US9637499, Compound 108)
Affinity DataIC50: 1.48E+3nMAssay Description:Inhibition of PDE4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed