BDBM142134 US8933079, 1.8

SMILES CN(C)Cc1ccc(C(=O)Cn2ccc(OCc3ccccc3)cc2=O)c(C)c1

InChI Key InChIKey=QONJYPHKWHUJOW-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 142134   

TargetMelanin-concentrating hormone receptor 1(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM142134(US8933079, 1.8)
Affinity DataIC50: 17nMpH: 7.0Assay Description:Membranes from CHO/Galpha16 cells stably transfected with human hMCH-1R are resuspended using a syringe (needle 0.6x25 mm) and diluted in test buffer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2015
Entry Details
Go to US Patent

TargetMelanin-concentrating hormone receptor 1(Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM142134(US8933079, 1.8)
Affinity DataIC50: 17nMAssay Description:Displacement of [125I]-MCH from human MCH-R1 expressed in CHO/Galpha16 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2016
Entry Details Article
PubMed