BDBM128302 US8796284, 13
SMILES CN(C)c1nc(nc(N)c1Br)-n1cccn1
InChI Key InChIKey=XFEJMGUHELBLFD-UHFFFAOYSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 128302
Affinity DataKi: 35nM ΔG°: -10.2kcal/moleT: 2°CAssay Description:Competition assays were carried out by incubation of membranes from hA1 receptors transfected to CHO cells, [3H]-DPCPX as radioligand, buffer (HEPES ...More data for this Ligand-Target Pair
Affinity DataKi: 50nM ΔG°: -10.4kcal/moleT: 2°CAssay Description:hese assays were performed at adenosine receptors transfected using a cAMP enzymeimmunoassay kit (Amersham Biosciences). CHO-A2A cells were seeded (1...More data for this Ligand-Target Pair