BDBM127937 US8796304, 2-([1,2,4]Triazolo[1,5-a]pyridin-2-ylsulfanylmethyl)-5H-imidazo[2,1-a]isoindole
SMILES C(Sc1nc2ccccn2n1)c1cn2Cc3ccccc3-c2n1
InChI Key InChIKey=NQTTXYWDJPGFTP-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 127937
Affinity DataIC50: 5.30E+3nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair