BDBM127924 US8796304, {2-[2-(5H-Imidazo[2,1-a]isoindol-2-yl)-ethyl]-5-methyl-[1,2,4]triazolo[1,5-a]pyrazin-8-yl}-methanol::US9062060, Table 1, Compound 5

SMILES Cc1cnc(CO)c2nc(CCc3cn4Cc5ccccc5-c4n3)nn12

InChI Key InChIKey=DVCBKKQNCIKRPU-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 127924   

LigandPNGBDBM127924(US8796304, {2-[2-(5H-Imidazo[2,1-a]isoindol-2-yl)-...)
Affinity DataIC50: 6.90nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM127924(US8796304, {2-[2-(5H-Imidazo[2,1-a]isoindol-2-yl)-...)
Affinity DataIC50: 6.90nMT: 2°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
In DepthDetails
US Patent