BDBM10144 lysine sulfonamide analogue 8

SMILES COC(=O)N1Cc2ccccc2C=C1C(=O)NCCCCC(CO)N(CC(C)C)S(=O)(=O)c1ccc(N)cc1

InChI Key InChIKey=KDTCSANVXICYGC-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 10144   

TargetDimer of Gag-Pol polyprotein [501-599](Human immunodeficiency virus type 1)
Ambrilia Biopharma

LigandPNGBDBM10144(lysine sulfonamide analogue 8)
Affinity DataIC50: 130nMpH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay. The proteolytic activity can be monitored by the increase in fluorescence in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed