BDBM50133817 4-(3-Chloro-pyridin-2-yl)-piperazine-1-carboxylic acid (4-tert-butyl-phenyl)-amide::BCTC::CHEMBL441472::N-(4-tert-butylphenyl)-4-(3-chloropyridin-2-yl)piperazine-1-carboxamide

SMILES CC(C)(C)c1ccc(NC(=O)N2CCN(CC2)c2ncccc2Cl)cc1

InChI Key InChIKey=ROGUAPYLUCHQGK-UHFFFAOYSA-N

Data  64 KI  39 IC50  1 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 104 hits for monomerid = 50133817   

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Tcg Lifesciences

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProtUniProtKB/TrEMBL
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TargetTransient receptor potential cation channel subfamily V member 1(Human)
Purdue Pharma

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 34nMAssay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in capsaicin-induced FLIPR assayMore data for this Ligand-Target Pair

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TargetTransient receptor potential cation channel subfamily V member 1(Human)
Purdue Pharma

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 30nMpH: 5.5Assay Description:Inhibition of human vanilloid receptor 1 in HEK293 cells in pH 5.5-induced FLIPR assayMore data for this Ligand-Target Pair

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UniProtKB/SwissProt
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TargetTransient receptor potential cation channel subfamily V member 1(Human)
Purdue Pharma

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 0.700nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells assessed as blockade of acid-induced receptor activation by [45Ca2+] uptake assayMore data for this Ligand-Target Pair

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UniProtKB/SwissProt
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TargetTransient receptor potential cation channel subfamily V member 1(Human)
Purdue Pharma

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 0.600nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as blockade of acid-induced receptor activation by FLIPR assayMore data for this Ligand-Target Pair

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UniProtKB/SwissProt
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TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Glaxosmithkline

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 0.600nMAssay Description:Antagonist activity at rat TRPV1 expressed in HEK293 cells assessed as blockade of acid-induced receptor activation by FLIPR assayMore data for this Ligand-Target Pair

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UniProtKB/SwissProt
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TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Glaxosmithkline

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 0.5nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as blockade of capsaicin-induced receptor activation by [45Ca2+] uptake assayMore data for this Ligand-Target Pair

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UniProtKB/SwissProt
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TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Glaxosmithkline

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 1.90nMAssay Description:Antagonist activity at rat TRPV1 expressed in HEK293 cells assessed as blockade of capsaicin-induced receptor activation by FLIPR assayMore data for this Ligand-Target Pair

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TargetTransient receptor potential cation channel subfamily V member 1(Human)
Purdue Pharma

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 5nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as blockade of capsaicin-induced receptor activation by FLIPR assayMore data for this Ligand-Target Pair

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TargetTransient receptor potential cation channel subfamily V member 1(Human)
Purdue Pharma

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 0.600nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells assessed as blockade of capsaicin-induced receptor activation by [45Ca2+] uptake assayMore data for this Ligand-Target Pair

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UniProtKB/SwissProt
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TargetTransient receptor potential cation channel subfamily V member 1(Human)
Purdue Pharma

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 5nMAssay Description:Antagonist activity at human recombinant TRPV1 expressed in human 1321N1 cells assessed as inhibition of capsaicin-induced calcium influx by FLIPR as...More data for this Ligand-Target Pair

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UniProtKB/SwissProt
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TargetTransient receptor potential cation channel subfamily A member 1(Human)
Sapienza University of Rome

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataEC50:  4.50E+3nMAssay Description:Antagonist activity at human TRPA1 expressed in HEK293 cells assessed as decrease in intracellular calcium levelMore data for this Ligand-Target Pair

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TargetTransient receptor potential cation channel subfamily V member 1(Human)
Purdue Pharma

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 6.70nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as decrease in intracellular calcium levelMore data for this Ligand-Target Pair

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TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Glaxosmithkline

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 35nMAssay Description:Vanilloid receptor subtype 1 antagonist activity based on its ability to block capsaicin-induced (CAP) activation of the rat VR1 channel in a HEK293 ...More data for this Ligand-Target Pair

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TargetTransient receptor potential cation channel subfamily V member 1(Human)
Purdue Pharma

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 0.180nMAssay Description:Antagonist activity against human TRPV1 expressed in T-REx HEK cells assessed as inhibition of capsaicin-induced increase in intracellular Ca2+ accum...More data for this Ligand-Target Pair

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UniProtKB/SwissProt
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TargetTransient receptor potential cation channel subfamily M member 8(Mouse)
University of Shizuoka

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 400nMAssay Description:Antagonist activity against mouse TRPM8 expressed in T-REx HEK cells assessed as inhibition of icilin-induced increase in intracellular Ca2+ accumula...More data for this Ligand-Target Pair

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TargetTransient receptor potential cation channel subfamily M member 8(Mouse)
University of Shizuoka

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 400nMAssay Description:Antagonist activity against mouse TRPM8 expressed in T-REx HEK cells assessed as inhibition of menthol-induced increase in intracellular Ca2+ accumul...More data for this Ligand-Target Pair

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TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Glaxosmithkline

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 0.700nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells assessed as blockade of acid-induced receptor activation by [45Ca2+] uptake assayMore data for this Ligand-Target Pair

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UniProtKB/SwissProt
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TargetTransient receptor potential cation channel subfamily M member 8(Rat)
University of Salerno

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 475nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as inhibition of menthol mediated current amplitude at +80 mV holding potential b...More data for this Ligand-Target Pair

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TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Sapienza University of Rome

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of FAAH-mediated hydrolysis of [3H]AEA in rat brain membraneMore data for this Ligand-Target Pair

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TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Glaxosmithkline

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 0.400nMAssay Description:Antagonist activity against capsaicin-induced 45calcium ion uptake in CHO cells expressing rat TRPV1More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
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TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Glaxosmithkline

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 0.5nMAssay Description:Antagonist activity against acid-induced 45calcium ion uptake in CHO cells expressing rat TRPV1 at pH5More data for this Ligand-Target Pair

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UniProtKB/SwissProt
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TargetTransient receptor potential cation channel subfamily V member 1(Human)
Purdue Pharma

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 35nMAssay Description:Inhibition of TRPV1 (unknown origin)More data for this Ligand-Target Pair

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TargetTransient receptor potential cation channel subfamily M member 8(Human)
Glenmark Pharmaceuticals

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 800nMAssay Description:Inhibition of TRPM8 (unknown origin)More data for this Ligand-Target Pair

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TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Glaxosmithkline

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 4.80nMAssay Description:Vanilloid receptor subtype 1 antagonist activity based on its ability to block low pH-induced activation of the rat VR1 channel in a HEK293 cell lineMore data for this Ligand-Target Pair

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TargetTransient receptor potential cation channel subfamily M member 8(Mouse)
University of Shizuoka

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 400nMAssay Description:Antagonist at TRPM8 isolated from mouse dorsal root ganglion cells expressed in HEK T-REx cells assessed as inhibition of icilin-induced intracellula...More data for this Ligand-Target Pair

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UniProtKB/SwissProt
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TargetTransient receptor potential cation channel subfamily M member 8(Mouse)
University of Shizuoka

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 350nMAssay Description:Antagonist at TRPM8 isolated from mouse dorsal root ganglion cells expressed in HEK T-REx cells assessed as inhibition of menthol-induced intracellul...More data for this Ligand-Target Pair

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TargetTransient receptor potential cation channel subfamily V member 1(Human)
Purdue Pharma

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 0.150nMAssay Description:Antagonist activity at human brain TRPV1 expressed in HEK293T cells assessed as inhibition of CAP-induced intracellular Ca2+ influx by fluorescence-b...More data for this Ligand-Target Pair

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TargetTransient receptor potential cation channel subfamily V member 1(Human)
Purdue Pharma

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 7nMAssay Description:Displacement of [3H]RTX from human TRPV1 expressed in HEK293 cell membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair

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TargetTransient receptor potential cation channel subfamily V member 1(Human)
Purdue Pharma

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 1.80nMAssay Description:Antagonist activity at recombinant human TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced activationMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
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TargetTransient receptor potential cation channel subfamily V member 1(Human)
Purdue Pharma

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 16nMAssay Description:Inhibition of human TRPV1 expressed in HEK293 cells assessed as reduction in capsaicin-induced activity pretreated for 2.5 mins followed by capsaicin...More data for this Ligand-Target Pair

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TargetTransient receptor potential cation channel subfamily V member 1(Human)
Purdue Pharma

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 9.60nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced intracellular calcium level preincubated for 2.5 mins followed by caps...More data for this Ligand-Target Pair

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TargetTransient receptor potential cation channel subfamily M member 8(Human)
Glenmark Pharmaceuticals

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 475nMAssay Description:Antagonist activity at TRPM8 (unknown origin) assessed as reduction in menthol-induced calcium influxMore data for this Ligand-Target Pair

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TargetTransient receptor potential cation channel subfamily V member 1(Human)
Purdue Pharma

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 19nMAssay Description:Antagonist activity at capsaicin-stimulated human TRPV1 receptor in aequorin expressing cells preincubated for 2.5 mins followed by capsaicin additio...More data for this Ligand-Target Pair

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TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Glaxosmithkline

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 4.90nMAssay Description:Antagonist activity at rat TRPV1 receptor expressed in HEK293T cells assessed as inhibition of capsaicin-induced calcium flux after 30 mins by Fluo-4...More data for this Ligand-Target Pair

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TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Glaxosmithkline

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at rat TRPV1 receptor expressed in HEK293T cells assessed as inhibition of temperature-induced calcium flux after 30 mins by Fluo...More data for this Ligand-Target Pair

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TargetTransient receptor potential cation channel subfamily V member 1(Human)
Purdue Pharma

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 19nMAssay Description:Antagonist activity at capsaicin-induced human recombinant TRPV1 expressed in CHO-K1 cells co-expressing aequorin incubated for 2.5 mins in presence ...More data for this Ligand-Target Pair

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TargetTransient receptor potential cation channel subfamily V member 1(Human)
Purdue Pharma

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 24nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced channel activationMore data for this Ligand-Target Pair

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TargetTransient receptor potential cation channel subfamily V member 1(Human)
Purdue Pharma

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 35nMAssay Description:Inhibition of TRPV1 (unknown origin)More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
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TargetTransient receptor potential cation channel subfamily V member 1(Human)
Purdue Pharma

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataIC50: 34nMAssay Description:Inhibition of human TRPV1More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchaseChEBI
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TargetMu-type opioid receptor(Rat)
Pudue Pharma Discovery Research

Curated by PDSP K_i Database

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataKi:  0.000950nMMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

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TargetTransient receptor potential cation channel subfamily V member 1(Human)
Purdue Pharma

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataKi:  2.5nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK cells assessed as inhibition of 10 nM capsaicin-induced calcium uptake by FLIPR assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchaseChEBI
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TargetTransient receptor potential cation channel subfamily V member 1(Human)
Purdue Pharma

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]RTX from human TRPV1 expressed in CHO cell membranes after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchaseChEBI
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TargetTransient receptor potential cation channel subfamily V member 1(Human)
Purdue Pharma

Curated by ChEMBL

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataKi:  11nMAssay Description:Displacement of [3H]MPOU from human TRPV1 expressed in CHO cell membranes after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
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TargetAcetylcholinesterase(Rat)
Pudue Pharma Discovery Research

Curated by PDSP K_i Database

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
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TargetAdenosine kinase(Rat)
Pudue Pharma Discovery Research

Curated by PDSP K_i Database

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

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TargetAlpha-1A adrenergic receptor(Rat)
Pudue Pharma Discovery Research

Curated by PDSP K_i Database

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

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TargetAlpha-2C adrenergic receptor(Rat)
Pudue Pharma Discovery Research

Curated by PDSP K_i Database

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

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TargetBeta-2 adrenergic receptor(Rat)
Pudue Pharma Discovery Research

Curated by PDSP K_i Database

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
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TargetType-1 angiotensin II receptor A(Rat)
Pudue Pharma Discovery Research

Curated by PDSP K_i Database

LigandBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)Copy SMILESCopy InChI

Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchaseChEBI
CHEMBLPC cidPC sidSimilars

In DepthDetails Article
Copy BDB DOIPubMed
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