BDBM50053173 (2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-1-ylmethyl-4-thia-1-aza-bicyclo[3.2.0]heptane-2-carboxylic acid::(2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-1-ylmethyl-4lambda 6-thia-1-aza-bicyclo[3.2.0]heptane-2-carboxylic acid::(2S,3S,5R)-3-methyl-4,4,7-trioxo-3-[1,2,3]triazol-1-ylmethyl-4lambda6-thia-1-aza-bicyclo[3.2.0]heptane-2-carboxylic acid::(2S,3S,5R)-3-methyl-7-oxo-3-(1H-1,2,3-triazol-1-ylmethyl)-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid 4,4-dioxide::3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-1-ylmethyl-4lambda*6*-thia-1-aza-bicyclo[3.2.0]heptane-2-carboxylic acid::CHEMBL404::CL-298741::TAZOBACTAM::US9120808, Tazobactam sodium salt::US9676777, TAZ::YTR-830H::Zosyn

SMILES C[C@]1(Cn2ccnn2)[C@@H](N2[C@@H](CC2=O)S1(=O)=O)C(O)=O

InChI Key InChIKey=LPQZKKCYTLCDGQ-UHFFFAOYSA-N

Data  4 KI  82 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 85 hits for monomerid = 50053173   

TargetBeta-lactamase OXA-1(Escherichia coli)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 4.80E+3nMAssay Description:Compound was tested for inhibition of Beta-lactamase from Bacteroides fragilis 36More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Enterobacter cloacae)
Lek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 1.81E+3nMAssay Description:Inhibition of Enterobacter cloacae AmpCMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Citrobacter gillenii)
Bicetre Hospital

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 40nMAssay Description:Inhibition of Citrobacter gillenii CIP 106783 Beta-lactamase GIL1 expressed in Escherichia coli DH10BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetallo-beta-lactamase L1 type 3(Pseudomonas maltophilia)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 4.00E+6nMAssay Description:Compound was tested for inhibition of Beta-lactamase from Xanthomonas maltophila 328More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Enterobacter cloacae)
Lek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 930nMAssay Description:Compound was tested for inhibition of Beta-lactamase from SHV-2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Citrobacter freundii)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 930nMAssay Description:Compound was tested for inhibition of Beta-lactamase from Citrobacter freundii 1982More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Escherichia coli (strain K12))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 1.80E+4nMAssay Description:Compound was tested for inhibition of Beta-lactamase from Escherichia coli SN03More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Morganella morganii)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 190nMAssay Description:Compound was tested for inhibition of beta-Lactamases from Morganell morgani U1627More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 2.11E+3nMAssay Description:Compound was tested for inhibition of Beta-lactamase from Pseudomonas aeruginosa GN10362More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetallo-beta-lactamase type 2(Bacteroides fragilis)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 1.00E+7nMAssay Description:Compound was tested for inhibition of Beta-lactamase from Bacteroides fragilis BF 101More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Bacillus licheniformis)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 510nMAssay Description:Compound was tested for inhibition of Beta-lactamase from Bacillus licheniformis 749/CMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase TEM(Escherichia coli)
Lek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 17nMAssay Description:Inhibition of Escherichia coli TEM1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Staphylococcus aureus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 500nMAssay Description:Compound was tested for inhibition of Beta-lactamase from Staphylococcus aureus PCIMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase TEM(Escherichia coli)
Lek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Escherichia coli WC3310 TEM-2More data for this Ligand-Target Pair
In DepthDetails Article

TargetBeta-lactamase(Enterobacter cloacae)
Lek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibitory activity against class C Beta-lactamase isolated from Enterobacter cloacaeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Pseudomonas aeruginosa (g-Proteobacteria))
The R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 60nMAssay Description:Inhibitory activity against class A Beta-lactamase TEM isolated from Enterobacter coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa beta-lactamase AmpC assessed as nitrocefin hydrolysis after 5 mins enzyme-compound preincubationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Enterobacter cloacae)
Lek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of Enterobacter cloacae beta-lactamase P99 assessed as nitrocefin hydrolysis after 5 mins enzyme-compound preincubationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Burkholderia cenocepacia)
H�Pital De Bic�Tre

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 500nMAssay Description:Inhibition of Burkholderia cenocepacia 07-34 beta-lactamase PenB1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Salmonella enterica subsp. enterica serovar Westha...)
Centre National De R£F£Rence Des Salmonella

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of Salmonella enterica serotype Westhampton beta-lactamase CTX-M-53More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Pseudomonas aeruginosa)
Hellenic Pasteur Institute

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 60nMAssay Description:Inhibition of Pseudomonas aeruginosa GES-13 beta lactamaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase OXA-1(Escherichia coli)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 432nMAssay Description:Inhibitory activity against Escherichia coli HA209 Class-V OXA-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails

TargetBeta-lactamase(Pseudomonas aeruginosa)
H�Pital De Bic�Tre

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa 51170 beta-lactamase BEL-1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Pseudomonas aeruginosa)
H�Pital De Bic�Tre

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa 531 beta-lactamase BEL-2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Pseudomonas luteola)
Institut Pasteur

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 40nMAssay Description:Inhibition of Pseudomonas luteola LAM Beta-lactamase LUT-1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Enterobacter cloacae)
Lek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 943nMAssay Description:Inhibitory activity against beta-Lactamase enzyme derived from Enterobacter cloacae P99More data for this Ligand-Target Pair
In DepthDetails Article

TargetBeta-lactamase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 950nMpH: 7.0Assay Description:For the measurement of β-lactamase inhibitory activity, 100 μM (final concentration) nitrocefin (Oxoid) was used as a substrate, and 2.5% D...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-lactamase BRO-1(Moraxella catarrhalis)TBA
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 33.3nMAssay Description:Inhibitory activity against Branhamella catarrhalis 89001 Class-III BRO-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails

TargetBeta-lactamase(Staphylococcus aureus)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 166nMAssay Description:Inhibitory activity against Staphylococcus aureus CJ8 beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails

TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against Proteus vulgaris HJ33C Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails

TargetBeta-lactamase(Klebsiella oxytoca)TBA
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 106nMAssay Description:Inhibitory activity against Klebsiella oxytoca HC7 Class-IV K1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails

TargetBeta-lactamase(Escherichia coli (strain K12))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 1.81E+3nMpH: 7.0 T: 2°CAssay Description:The inhibitory concentrations (IC50, [uM]) of the beta -lactamase inhibitors against purified TEM-1, SHV-1 and AmpC beta -lactamases are assessed by ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetBeta-lactamase SHV-1(Pseudomonas aeruginosa (g-Proteobacteria))TBA
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 133nMAssay Description:Inhibitory activity against Escherichia coli HA208 Class-III SHV-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails

TargetBeta-lactamase(Enterobacter cloacae)
Lek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 333nMAssay Description:Inhibitory activity against Enterobacter cloacae HC8 Class-I beta-lactamase enzyme type P99More data for this Ligand-Target Pair
In DepthDetails

TargetBeta-lactamase TEM(Escherichia coli)
Lek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against Escherichia coli HA58R Class-III TEM-1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails

TargetBeta-lactamase(Citrobacter freundii)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 166nMAssay Description:Inhibitory activity against Citrobacter freundii 87470 Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails

TargetMetallo-beta-lactamase type 2(Bacteroides fragilis)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 2.66E+3nMAssay Description:Inhibitory activity against Bacteroides fragilis 88854 Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails

TargetBeta-lactamase TEM(Escherichia coli)
Lek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 90nMAssay Description:Inhibition of Escherichia coli K12 TEM1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Escherichia coli)
Institut Pasteur Hellenique

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 10nMAssay Description:Inhibition of Escherichia coli beta-lactamase SCO1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetClass A beta-lactamase BCL-1(Bacillus clausii)
H�Pital De Bic�Tre

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 4nMAssay Description:Inhibition of Bacillus clausii NR beta-lactamase BCL1 expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase SHV-1(Pseudomonas aeruginosa (g-Proteobacteria))TBA
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 222nMAssay Description:Inhibition of Escherichia coli SHV1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 820nMAssay Description:Compound was tested for inhibition of Beta-lactamase from Pseudomonas aeruginosa 18SHMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Enterobacter cloacae)
Lek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 4.80E+4nMAssay Description:In vitro inhibitory activity against Beta-lactamase AmpC of class C enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Escherichia coli (strain K12))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 250nMAssay Description:Inhibitory activity against class A TEM-1 beta-lactamaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Enterobacter cloacae)
Lek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 1.02E+5nMAssay Description:Inhibitory activity against Class C beta-lactamaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMetallo-beta-lactamase type 2(Bacteroides fragilis)
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro inhibitory concentration against CCRA enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Escherichia coli (strain K12))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 4.80E+4nMAssay Description:In vitro inhibitory concentration against AmpC enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase TEM(Escherichia coli)
Lek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 60nMAssay Description:In vitro inhibitory concentration against TEM-1 enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Enterobacter cloacae)
Lek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 8.50E+4nMAssay Description:Compound was tested for inhibition of Beta-lactamase from Ent. cloacae 6300More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-lactamase(Escherichia coli (strain K12))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50: 9.80E+4nMAssay Description:Compound was tested for inhibition of Beta-lactamase from Bacteroides fragilis 98More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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