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15 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Prodrugs of purine and pyrimidine analogues for the intestinal di/tri-peptide transporter PepT1: affinity for hPepT1 in Caco-2 cells, drug release in aqueous media and in vitro metabolism.EBI
The Royal Danish School of Pharmacy
Novel class of potent 4-arylalkyl substituted 3-isoxazolol GABA(A) antagonists: synthesis, pharmacology, and molecular modeling.EBI
The Royal Danish School of Pharmacy
Ligands for glutamate receptors: design and therapeutic prospects.EBI
The Royal Danish School of Pharmacy
Solid-phase synthesis of polyamine toxin analogues: potent and selective antagonists of Ca2+-permeable AMPA receptors.EBI
The Royal Danish School of Pharmacy
Selective agonists at group II metabotropic glutamate receptors: synthesis, stereochemistry, and molecular pharmacology of (S)- and (R)-2-amino-4-(4-hydroxy[1,2,5]thiadiazol-3-yl)butyric acid.EBI
The Royal Danish School of Pharmacy
Solid-phase synthesis and pharmacological evaluation of analogues of PhTX-12-A potent and selective nicotinic acetylcholine receptor antagonist.EBI
The Royal Danish School of Pharmacy
Selective antagonists at group I metabotropic glutamate receptors: synthesis and molecular pharmacology of 4-aryl-3-isoxazolol amino acids.EBI
The Royal Danish School of Pharmacy
Novel 1-hydroxyazole bioisosteres of glutamic acid. Synthesis, protolytic properties, and pharmacology.EBI
The Royal Danish School of Pharmacy
A new concept for multidimensional selection of ligand conformations (MultiSelect) and multidimensional scoring (MultiScore) of protein-ligand binding affinities.EBI
The Royal Danish School of Pharmacy
Bioisosteric determinants for subtype selectivity of ligands for heteromeric GABA(A) receptors.EBI
The Royal Danish School of Pharmacy
Synthesis and pharmacology of the baclofen homologues 5-amino-4-(4-chlorophenyl)pentanoic acid and the R- and S-enantiomers of 5-amino-3-(4-chlorophenyl)pentanoic acid.EBI
The Royal Danish School of Pharmacy
Solid-phase synthesis and biological evaluation of a combinatorial library of philanthotoxin analogues.EBI
The Royal Danish School of Pharmacy
Piperidin-4-yl azetidine derivatives as JAK1 inhibitorsBDB
Incyte Holdings
Dual acting norepinephrine reuptake inhibitors and 5-HT(2A) receptor antagonists: Identification, synthesis and activity of novel 4-aminoethyl-3-(phenylsulfonyl)-1H-indoles.BDB
Wyeth Research