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37 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Solution-phase microwave assisted parallel synthesis, biological evaluation and in silico docking studies of N,N'-disubstituted thioureas derived from 3-chlorobenzoic acid.EBI
Quaid-I-Azam University
Synthesis of potent urease inhibitors based on disulfide scaffold and their molecular docking studies.EBI
Universiti Teknologi Mara (Uitm)
Discovery of indole-based tetraarylimidazoles as potent inhibitors of urease with low antilipoxygenase activity.EBI
University of The Punjab
Design and synthesis of new barbituric- and thiobarbituric acid derivatives as potent urease inhibitors: Structure activity relationship and molecular modeling studies.EBI
The Islamia University of Bahawalpur
Synthesis of novel derivatives of oxindole, their urease inhibition and molecular docking studies.EBI
Universiti Teknologi Mara Puncak Alam Campus
Implications of N-capped urea/thiourea and C-capped 3-(1-piperazinyl)-1,2-benzisothiazole with bridging Gly-Val/Phe-Gly-Val-Pro as therapeutic targets.EBI
University of Mysore
Synthesis and in vitro urease inhibitory activity of N,N'-disubstituted thioureas.EBI
University Karachi
Solution-phase microwave assisted parallel synthesis of N,N'-disubstituted thioureas derived from benzoic acid: biological evaluation and molecular docking studies.EBI
Quaid-I-Azam University
3D-QSAR CoMFA studies on bis-coumarine analogues as urease inhibitors: a strategic design in anti-urease agents.EBI
University of Karachi
Synthesis, biological assay in vitro and molecular docking studies of new Schiff base derivatives as potential urease inhibitors.EBI
Comsats Institute of Information Technology
Synthesis, antioxidant activities and urease inhibition of some new 1,2,4-triazole and 1,3,4-thiadiazole derivatives.EBI
Quaid-I-Azam University
Bioactive oligostilbenoids from the stem bark of Hopea exalata.EBI
Nanjing University
Facile one-pot synthesis of thio and selenourea derivatives: a new class of potent urease inhibitors.EBI
Institute of Science
Insights into the recent progress in the medicinal chemistry of pyranopyrimidine analogs.EBI
Mansoura University
Developing new hybrid scaffold for urease inhibition based on carbazole-chalcone conjugates: Synthesis, assessment of therapeutic potential and computational docking analysis.EBI
Quaid-I-Azam University
Synthesis and urease inhibitory potential of benzophenone sulfonamide hybrid in vitro and in silico.EBI
University of Karachi
1,2,3-Triazole-containing hybrids as leads in medicinal chemistry: A recent overview.EBI
Chinese Academy of Sciences
Rational approaches, design strategies, structure activity relationship and mechanistic insights for therapeutic coumarin hybrids.EBI
Guru Nanak Dev University
Design, synthesis and biological activities of some 7-aminocephalosporanic acid derivatives.EBI
Karadeniz Technical University
Microwave assisted synthesis of some hybrid molecules derived from norfloxacin and investigation of their biological activities.EBI
Karadeniz Technical University
Bisindolylmethane thiosemicarbazides as potential inhibitors of urease: Synthesis and molecular modeling studies.EBI
Imam Abdulrahman Bin Faisal University
Synthesis and molecular docking study of some 5,6-dichloro-2-cyclopropyl-1H-benzimidazole derivatives bearing triazole, oxadiazole, and imine functionalities as potent inhibitors of urease.EBI
Recep Tayyip Erdogan University
Substituted pyrimidine compounds and their use as SYK inhibitorsBDB
Genosco
Non-peptide macrocyclic histone deacetylese (HDAC) inhibitors and methods of making and using thereofBDB
Georgia Tech Research
Azaspirodecanone compoundsBDB
Hoffmann-La Roche
Pyrazol-4-yl-heterocyclyl-carboxamide compounds and methods of useBDB
F. Hoffmann-La Roche
Imidazo pyrazinesBDB
Hoffmann-La Roche
Dihydrooxazol-2-amine derivativesBDB
Hoffmann-La Roche
Functional selectivity of dopamine receptor agonists. I. Selective activation of postsynaptic dopamine D2 receptors linked to adenylate cyclase.BDB
University of North Carolina
Synthesis and in vitro opioid activity profiles of DALDA analogues.BDB
Clinical Research Institute of Montreal
Behaviroal, pharmacological, and molecular characterization of an amphibian cannabinoid receptor.BDB
Oregon State University
Glucose-based spiro-isoxazolines: a new family of potent glycogen phosphorylase inhibitors.BDB
Universite De Lyon