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24 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Novel PARP7 Inhibitors for Treating Cancer.EBI
Smith, Gambrell & Russell
Discovery of Quinazoline-2,4(1EBI
Chinese Academy of Medical Sciences and Peking Union Medical College
PARP7 Inhibition: A Promising Pathway to Advancements in Cancer Therapy.EBI
Usona Institute
YCH1899, a Highly Effective Phthalazin-1(2EBI
Shanghai Institute of Materia Medica
[1,2,4]Triazolo[3,4-EBI
University of Oulu
Discovery of the Potent and Highly Selective PARP7 Inhibitor as a Novel Immunotherapeutic Agent for Tumors.EBI
China Pharmaceutical University
Optimization of a Screening Hit toward M2912, an Oral Tankyrase Inhibitor with Antitumor Activity in Colorectal Cancer Models.EBI
Merck
Recent Discovery of PARP7 Inhibitors as Anticancer Agents.EBI
Usona Institute
Medicinal Chemistry Perspective on Targeting Mono-ADP-Ribosylating PARPs with Small Molecules.EBI
University of Perugia
Rational design, synthesis and biological evaluation of dual PARP-1/2 and TNKS1/2 inhibitors for cancer therapy.EBI
Nanjing University
Potent 2,3-dihydrophthalazine-1,4-dione derivatives as dual inhibitors for mono-ADP-ribosyltransferases PARP10 and PARP15.EBI
University of Perugia
Discovery of Pamiparib (BGB-290), a Potent and Selective Poly (ADP-ribose) Polymerase (PARP) Inhibitor in Clinical Development.EBI
TBA
Discovery and Optimization of 2-Arylquinazolin-4-ones into a Potent and Selective Tankyrase Inhibitor Modulating Wnt Pathway Activity.EBI
Merck Healthcare
Rational Design of Cell-Active Inhibitors of PARP10.EBI
Oregon Health and Science University
SHP2 phosphatase allosteric inhibitorBDB
Beijing Shenogen Pharma Group
HETEROBIVALENT AND HOMOBIVALENT AGENTS TARGETING FIBROBLAST ACTIVATION PROTEIN ALPHA AND/OR PROSTATE-SPECIFIC MEMBRANE ANTIGENBDB
The Johns Hopkins University
3-phenoxyazetidin-1-yl-heteroaryl pyrrolidine derivatives and the use thereof as medicamentBDB
Boehringer Ingelheim International
NOVEL COMPOUNDS, COMPOSITIONS, AND THERAPEUTIC USES THEREOFBDB
Breakpoint Therapeutics
COMPOUNDS AND RADIOLIGANDS FOR TARGETING NEUROTENSIN RECEPTOR AND USES THEREOFBDB
Full-Life Technologies HK
CYCLIN-DEPENDENT KINASE INHIBITING COMPOUNDS FOR THE TREATMENT OF MEDICAL DISORDERSBDB
G1 Therapeutics
Compounds useful as RET inhibitorsBDB
Cancer Research Technology
Methods of inhibiting kinasesBDB
Insilico Medicine Ip
Pteridine dione monocarboxylate transporter inhibitorsBDB
The Scripps Research Institute
Compounds as indoleamine 2,3-dioxygenase inhibitorsBDB
Merck Sharp & Dohme