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20 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Discovery of Selective Small Molecule Inhibitors of Monoacylglycerol Acyltransferase 3.EBI
Pfizer
Discovery of a Novel Series of N-Phenylindoline-5-sulfonamide Derivatives as Potent, Selective, and Orally Bioavailable Acyl CoA:Monoacylglycerol Acyltransferase-2 Inhibitors.EBI
Takeda Pharmaceutical
Identification and design of a novel series of MGAT2 inhibitors.EBI
Astrazeneca
Design of Next-Generation DGAT2 Inhibitor PF-07202954 with Longer Predicted Half-Life.EBI
Pfizer
Discovery of EBI
TBA
Discovery of Ervogastat (PF-06865571): A Potent and Selective Inhibitor of Diacylglycerol Acyltransferase 2 for the Treatment of Non-alcoholic Steatohepatitis.EBI
Pfizer
Screening Hit to Clinical Candidate: Discovery of BMS-963272, a Potent, Selective MGAT2 Inhibitor for the Treatment of Metabolic Disorders.EBI
TBA
Monoacylglycerol Acyltransferase 2 (MGAT2) Inhibitors for the Treatment of Metabolic Diseases and Nonalcoholic Steatohepatitis (NASH).EBI
TBA
Discovery and Pharmacology of a Novel Class of Diacylglycerol Acyltransferase 2 Inhibitors.EBI
Merck
PHTHALAZINE DERIVATIVES AS PYRUVATE KINASE MODULATORSBDB
Sitryx Therapeutics
ARYL HETEROCYCLIC COMPOUNDS AS Kv1.3 POTASSIUM SHAKER CHANNEL BLOCKERSBDB
D.E. Shaw Research
Substituted amino acids as integrin inhibitorsBDB
Pliant Therapeutics
Substituted imidazopyridazinesBDB
Bayer Pharma Aktiengesellschaft
Substituted benzoxazolesBDB
Bayer Pharma Aktiengesellschaft
Structural basis of pharmacological chaperoning for human ß-galactosidase.BDB
The University of Tokyo
Synthesis and pharmacological characterization of novel xanthine carboxylate amides as A2A adenosine receptor ligands exhibiting bronchospasmolytic activity.BDB
Panjab University
Cyclic ether DGAT1 inhibitorscyclic ether DGAT1 inhibitorsBDB
Novartis
Phenoxyethoxy compoundsBDB
Eli Lilly
Prokineticin receptor antagonists and uses thereofBDB
University of California
Type II Ligands as Chemical Auxiliaries To Favor Enzymatic Transformations by P450 2E1.BDB
Mcgill University