PMID

Data

Article Title

Organization

Synthesis and biological evaluation of a unique heparin mimetic hexasaccharide for structure-activity relationship studies.

Momenta Pharmaceuticals

Structure-kinetic relationships--an overlooked parameter in hit-to-lead optimization: a case of cyclopentylamines as chemokine receptor 2 antagonists.

Leiden University

Fragment-based discovery of 6-substituted isoquinolin-1-amine based ROCK-I inhibitors.

Msd

Identification and Optimization of a Ligand-Efficient Benzoazepinone Bromodomain and Extra Terminal (BET) Family Acetyl-Lysine Mimetic into the Oral Candidate Quality Molecule I-BET432.

Gsk

Design, Synthesis, and Characterization of I-BET567, a Pan-Bromodomain and Extra Terminal (BET) Bromodomain Oral Candidate.

Glaxosmithkline R&D

Heparan Sulfate Mimetics Differentially Affect Homologous Chemokines and Attenuate Cancer Development.

Indian Institute of Science Education and Research