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10 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
2-(3-Methoxyphenyl)quinazoline Derivatives: A New Class of Direct Constitutive Androstane Receptor (CAR) Agonists.EBI
Palacky University In Olomouc
Development of CINPA1 analogs as novel and potent inverse agonists of constitutive androstane receptor.EBI
St. Jude Children'S Research Hospital
Identification of the first inverse agonist of retinoid-related orphan receptor (ROR) with dual selectivity for RORß and ROR¿t.EBI
Phenex Pharmaceuticals
Synthesis and pharmacological validation of a novel series of non-steroidal FXR agonists.EBI
Phenex Pharmaceuticals
Discovery of Novel Human Constitutive Androstane Receptor Agonists with the Imidazo[1,2-EBI
Czech Academy of Sciences
GNE-235: A Lead Compound Selective for the Second Bromodomain of PBRM1.EBI
Genentech
Discovery of 3α,7α,11β-Trihydroxy-6α-ethyl-5β-cholan-24-oic Acid (TC-100), a Novel Bile Acid as Potent and Highly Selective FXR Agonist for Enterohepatic Disorders.EBI
Tes Pharma
Tuning Nuclear Receptor Selectivity of Wy14,643 towards Selective Retinoid X Receptor Modulation.EBI
Goethe University Frankfurt
DL5050, a Selective Agonist for the Human Constitutive Androstane Receptor.EBI
University of Maryland
Human constitutive androstane receptor agonist DL5016: A novel sensitizer for cyclophosphamide-based chemotherapies.EBI
University of Maryland