PMID

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Article Title

Organization

Discovery and structural modification of inhibitors of methionine aminopeptidases from Escherichia coli and Saccharomyces cerevisiae.

Chinese Academy of Sciences

Inhibition of monometalated methionine aminopeptidase: inhibitor discovery and crystallographic analysis.

University of Kansas

Metal-mediated inhibition of Escherichia coli methionine aminopeptidase: structure-activity relationships and development of a novel scoring function for metal-ligand interactions.

Saarland University

Metalloform-selective inhibition: synthesis and structure-activity analysis of Mn(II)-form-selective inhibitors of Escherichia coli methionine aminopeptidase.

Graduate School of Chinese Academy of Sciences

Identification of potent type I MetAPs inhibitors by simple bioisosteric replacement. Part 2: SAR studies of 5-heteroalkyl substituted TCAT derivatives.

Shanghai Graduate School of The Chinese Academy of Sciences

Identification of potent type I MetAP inhibitors by simple bioisosteric replacement. Part 1: Synthesis and preliminary SAR studies of thiazole-4-carboxylic acid thiazol-2-ylamide derivatives.

Graduate School of The Chinese Academy of Sciences

Inhibitors of type I MetAPs containing pyridine-2-carboxylic acid thiazol-2-ylamide. Part 1: SAR studies on the determination of the key scaffold.

Chinese Academy of Sciences

Beta-aminoketones as prodrugs for selective irreversible inhibitors of type-1 methionine aminopeptidases.

Heidelberg University

Serendipitous discovery of novel bacterial methionine aminopeptidase inhibitors.

The Procter & Gamble Pharmaceuticals