PMID

Data

Article Title

Organization

Short Hydrophobic Peptides with Cyclic Constraints Are Potent Glucagon-like Peptide-1 Receptor (GLP-1R) Agonists.

University of Queensland

Peptide inhibitors of the Escherichia coli DsbA oxidative machinery essential for bacterial virulence.

University of Queensland

Structure aided design of chimeric antibiotics.

University of Queensland

Conformational selection of inhibitors and substrates by proteolytic enzymes: implications for drug design and polypeptide processing.

University of Queensland

Protease inhibitors: current status and future prospects.

University of Queensland

Inhibition of S/G2 phase CDK4 reduces mitotic fidelity.

University of Queensland

Antimalarial activity of azadipeptide nitriles.

University of Queensland

Molecular engineering of conotoxins: the importance of loop size to alpha-conotoxin structure and function.

University of Queensland

Synthesis and in vitro evaluation of a library of modified endomorphin 1 peptides.

University of Queensland

Internalisation of the mu-opioid receptor by endomorphin-1 and leu-enkephalin is dependant on aromatic amino acid residues.

University of Queensland

Profiling the enzymatic properties and inhibition of human complement factor B.

University of Queensland

Enzyme adaptation to inhibitor binding: a cryptic binding site in phenylethanolamine N-methyltransferase.

University of Queensland

Antiproliferative and phenotype-transforming antitumor agents derived from cysteine.

University of Queensland

Hormone-like conopeptides - new tools for pharmaceutical design.

University of Queensland

Determining the necessity of phenyl ring π-character in warfarin.

University of Queensland

Low-molecular-weight peptidic and cyclic antagonists of the receptor for the complement factor C5a.

University of Queensland

Small molecular probes for G-protein-coupled C5a receptors: conformationally constrained antagonists derived from the C terminus of the human plasma protein C5a.

University of Queensland

Herbicide-binding sites revealed in the structure of plant acetohydroxyacid synthase.

University of Queensland

A refined agonist pharmacophore for protease activated receptor 2.

University of Queensland

Cyclic MrIA: a stable and potent cyclic conotoxin with a novel topological fold that targets the norepinephrine transporter.

University of Queensland

Fused bicyclic pyrimidine derivatives and uses thereof

University of Colorado

BENZODIAZEPINE DERIVATIVES USEFUL IN TREATING A RESPIRATORY SYNCYTIAL VIRUS INFECTION

Reviral

Thiazoles as modulators of RORγt

Janssen Pharmaceutica

Unexpected novel binding mode of pyrrolidine-based aspartyl protease inhibitors: design, synthesis and crystal structure in complex with HIV protease.

Philipps-Universität Marburg

Multisubstituted aromatic compounds as serine protease inhibitors

Verseon

Dihydropyrancarboxamides related to zanamivir: a new series of inhibitors of influenza virus sialidases. 1. Discovery, synthesis, biological activity, and structure-activity relationships of 4-guanidino- and 4-amino-4H-pyran-6-carboxamides.

Glaxo Wellcome Research and Development