PMID

Data

Article Title

Organization

Novel 3-Substituted 7-Phenylpyrrolo[3,2-f]quinolin-9(6H)-ones as Single Entities with Multitarget Antiproliferative Activity.

University of Padova

Novel 9'-substituted-noscapines: synthesis with Suzuki cross-coupling, structure elucidation and biological evaluation.

University of Padova

Discovery of biarylaminoquinazolines as novel tubulin polymerization inhibitors.

University of Padova

Design, synthesis, and structure-activity relationships of azolylmethylpyrroloquinolines as nonsteroidal aromatase inhibitors.

University of Padova

Quinazoline-based multi-tyrosine kinase inhibitors: synthesis, modeling, antitumor and antiangiogenic properties.

University of Padova

Psoralen derivatives as inhibitors of NF-¿B/DNA interaction: synthesis, molecular modeling, 3D-QSAR, and biological evaluation.

University of Padova

8-Hydroxynaphthalene-1,4-dione derivative as novel compound for glioma treatment.

University of Padova

Hypericins and thioredoxin reductase: Biochemical and docking studies disclose the molecular basis for effective inhibition by naphthodianthrones.

University of Padova

Side chain cyclization based on serine residues: synthesis, structure, and activity of a novel cyclic analogue of the parathyroid hormone fragment 1-11.

University of Padova

Combining selectivity and affinity predictions using an integrated Support Vector Machine (SVM) approach: An alternative tool to discriminate between the human adenosine A(2A) and A(3) receptor pyrazolo-triazolo-pyrimidine antagonists binding sites.

University of Padova

Anthracene based compounds as new L-type Ca2+ channel blockers: design, synthesis, and full biological profile.

University of Padova

Aminoacyl-anthraquinone conjugates as telomerase inhibitors: synthesis, biophysical and biological evaluation.

University of Padova

Tri-, tetra- and heptacyclic perylene analogues as new potential antineoplastic agents based on DNA telomerase inhibition.

University of Padova

Scaffold Repurposing of in-House Chemical Library toward the Identification of New Casein Kinase 1 δ Inhibitors.

University of Padova

Third-generation CDK inhibitors: A review on the synthesis and binding modes of Palbociclib, Ribociclib and Abemaciclib.

University of Padova

Evaluating the effects of fluorine on biological properties and metabolic stability of some antitubulin 3-substituted 7-phenyl-pyrroloquinolinones.

University of Padova

Novel polyamine analogues: from substrates towards potential inhibitors of monoamine oxidases.

University of Padova

Targeting RORs nuclear receptors by novel synthetic steroidal inverse agonists for autoimmune disorders.

University of Padova

Substituted quinazoline compounds and preparation and uses thereof

Sunshine Lake Pharma

Histone demethylase inhibitors

Celgene Quanticel Research

Synthesis and anti-HIV-1 activity of a series of imidazo[1,5-b]pyridazines.

Glaxo Group Research