The first public molecular recognition database, BindingDB supports research, education and practice in drug discovery, pharmacology and related fields.

BindingDB contains 3.0M data for 1.3M Compounds and 9.6K Targets. Of those, 1.5M data for 695K Compounds and 4.7K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

If BindingDB was of value to your research, please take a moment to donate to this nonprofit project. Your donation will let us provide you with more data and improved service.

Advanced Search

150 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
3-Hydroxy-1H-quinazoline-2,4-dione as a New Scaffold To Develop Potent and Selective Inhibitors of the Tumor-Associated Carbonic Anhydrases IX and XII.EBI
Universita Degli Studi Di Firenze
The 1,2,4-Triazolo[4,3-a]pyrazin-3-one as a Versatile Scaffold for the Design of Potent Adenosine Human Receptor Antagonists. Structural Investigations to Target the AEBI
Universita Degli Studi Di Firenze
Lead Development of Thiazolylsulfonamides with Carbonic Anhydrase Inhibitory Action.EBI
Universita Degli Studi Di Firenze
Design, Synthesis, and Pharmacological Characterization of 2-(2-Furanyl)thiazolo[5,4-d]pyrimidine-5,7-diamine Derivatives: New Highly Potent AEBI
Universita Degli Studi Di Firenze
Dithiocarbamates effectively inhibit theß-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa.EBI
Universita Degli Studi Di Firenze
Coumarins and other fused bicyclic heterocycles with selective tumor-associated carbonic anhydrase isoforms inhibitory activity.EBI
Universita Degli Studi Di Firenze
Benzenesulfonamides Incorporating Flexible Triazole Moieties Are Highly Effective Carbonic Anhydrase Inhibitors: Synthesis and Kinetic, Crystallographic, Computational, and Intraocular Pressure Lowering Investigations.EBI
Universita Degli Studi Di Firenze
Synthesis 4-[2-(2-mercapto-4-oxo-4H-quinazolin-3-yl)-ethyl]-benzenesulfonamides with subnanomolar carbonic anhydrase II and XII inhibitory properties.EBI
Universita Degli Studi Di Firenze
Bortezomib inhibits bacterial and fungalß-carbonic anhydrases.EBI
Universita Degli Studi Di Firenze
N-Nitrosulfonamides: A new chemotype for carbonic anhydrase inhibition.EBI
Universita Degli Studi Di Firenze
Kinetic and X-ray crystallographic investigations of substituted 2-thio-6-oxo-1,6-dihydropyrimidine-benzenesulfonamides acting as carbonic anhydrase inhibitors.EBI
Universita Degli Studi Di Firenze
Exploring the 2- and 5-positions of the pyrazolo[4,3-d]pyrimidin-7-amino scaffold to target human A1 and A2A adenosine receptors.EBI
Universita Degli Studi Di Firenze
Comparison of the sulfonamide inhibition profiles of thea-,ß- and¿-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae.EBI
Universita Degli Studi Di Firenze
Anion inhibition studies of theß-carbonic anhydrase from the pathogenic bacterium Vibrio cholerae.EBI
Universita Degli Studi Di Firenze
Sulfonamide inhibition studies of the¿-carbonic anhydrase from the Antarctic bacterium Colwellia psychrerythraea.EBI
Universita Degli Studi Di Firenze
Sulfonamide inhibition studies of theß-carbonic anhydrase from the pathogenic bacterium Vibrio cholerae.EBI
Universita Degli Studi Di Firenze
Thioxocoumarins Show an Alternative Carbonic Anhydrase Inhibition Mechanism Compared to Coumarins.EBI
Universita Degli Studi Di Firenze
Structural refinement of pyrazolo[4,3-d]pyrimidine derivatives to obtain highly potent and selective antagonists for the human A3 adenosine receptor.EBI
Universita Degli Studi Di Firenze
Sulfonamide inhibition studies of thea-carbonic anhydrase from the gammaproteobacterium Thiomicrospira crunogena XCL-2, TcruCA.EBI
Universita Degli Studi Di Firenze
Inhibition of mammalian carbonic anhydrase isoforms I-XIV with a series of phenolic acid esters.EBI
Universita Degli Studi Di Firenze
Click-tailed coumarins with potent and selective inhibitory action against the tumor-associated carbonic anhydrases IX and XII.EBI
Universita Degli Studi Di Firenze
Cyclodextrin complexation highly enhances efficacy of arylsulfonylureido benzenesulfonamide carbonic anhydrase inhibitors as a topical antiglaucoma agents.EBI
Universita Degli Studi Di Firenze
Sulfonamide inhibition studies of the¿-carbonic anhydrase from the Antarctic bacterium Pseudoalteromonas haloplanktis.EBI
Universita Degli Studi Di Firenze
Inhibition studies of bacterial, fungal and protozoanß-class carbonic anhydrases with Schiff bases incorporating sulfonamide moieties.EBI
Universita Degli Studi Di Firenze
Anion inhibition study of theß-class carbonic anhydrase (PgiCAb) from the oral pathogen Porphyromonas gingivalis.EBI
Universita Degli Studi Di Firenze
a-Carbonic Anhydrases Possess Thioesterase Activity.EBI
Universita Degli Studi Di Firenze
Synthesis of a new series of dithiocarbamates with effective human carbonic anhydrase inhibitory activity and antiglaucoma action.EBI
Universita Degli Studi Di Firenze
A class of sulfonamide carbonic anhydrase inhibitors with neuropathic pain modulating effects.EBI
Universita Degli Studi Di Firenze
Sulfonamide inhibition studies of the¿-class carbonic anhydrase from the malaria pathogen Plasmodium falciparum.EBI
Universita Degli Studi Di Firenze
Sulfonamides with Potent Inhibitory Action and Selectivity against thea-Carbonic Anhydrase from Vibrio cholerae.EBI
Universita Degli Studi Di Firenze
Synthesis of sulfonamides with effective inhibitory action against Porphyromonas gingivalis¿-carbonic anhydrase.EBI
Universita Degli Studi Di Firenze
Further studies on pyrazolo[1',5':1,6]pyrimido[4,5-d]pyridazin-4(3H)-ones as potent and selective human A1 adenosine receptor antagonists.EBI
Universita Degli Studi Di Firenze
A class of 4-sulfamoylphenyl-¿-aminoalkyl ethers with effective carbonic anhydrase inhibitory action and antiglaucoma effects.EBI
Universita Degli Studi Di Firenze
Structural insights on carbonic anhydrase inhibitory action, isoform selectivity, and potency of sulfonamides and coumarins incorporating arylsulfonylureido groups.EBI
Universita Degli Studi Di Firenze
Inhibition of carbonic anhydrase isoforms I, II, IX and XII with novel Schiff bases: identification of selective inhibitors for the tumor-associated isoforms over the cytosolic ones.EBI
Universita Degli Studi Di Firenze
Xanthates and trithiocarbonates strongly inhibit carbonic anhydrases and show antiglaucoma effects in vivo.EBI
Universita Degli Studi Di Firenze
The alpha-carbonic anhydrase from the thermophilic bacterium Sulfurihydrogenibium yellowstonense YO3AOP1 is highly susceptible to inhibition by sulfonamides.EBI
Universita Degli Studi Di Firenze
Sulfonamide inhibition studies of thed-carbonic anhydrase from the diatom Thalassiosira weissflogii.EBI
Universita Degli Studi Di Firenze
Anion inhibition studies of aß-carbonic anhydrase from Clostridium perfringens.EBI
Universita Degli Studi Di Firenze
Optimization of N-benzoylindazole derivatives as inhibitors of human neutrophil elastase.EBI
Universita Degli Studi Di Firenze
Further studies on 2-arylacetamide pyridazin-3(2H)-ones: design, synthesis and evaluation of 4,6-disubstituted analogs as formyl peptide receptors (FPRs) agonists.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors: inhibition of theß-class enzyme from the pathogenic yeast Candida glabrata with sulfonamides, sulfamates and sulfamides.EBI
Universita Degli Studi Di Firenze
Anion inhibition studies of thea-carbonic anhydrase from the pathogenic bacterium Vibrio cholerae.EBI
Universita Degli Studi Di Firenze
Mono-/dihydroxybenzoic acid esters and phenol pyridinium derivatives as inhibitors of the mammalian carbonic anhydrase isoforms I, II, VII, IX, XII and XIV.EBI
Universita Degli Studi Di Firenze
Novel small molecule protein arginine deiminase 4 (PAD4) inhibitors.EBI
Universita Degli Studi Di Firenze
Anion inhibition studies of the fastest carbonic anhydrase (CA) known, the extremo-CA from the bacterium Sulfurihydrogenibium azorense.EBI
Universita Degli Studi Di Firenze
Dithiocarbamates strongly inhibit carbonic anhydrases and show antiglaucoma action in vivo.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors. Antioxidant polyphenols effectively inhibit mammalian isoforms I-XV.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors. Inhibition of mammalian isoforms I-XIV with a series of natural product polyphenols and phenolic acids.EBI
Universita Degli Studi Di Firenze
Deciphering the mechanism of carbonic anhydrase inhibition with coumarins and thiocoumarins.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors. Inhibition of the Rv1284 and Rv3273 beta-carbonic anhydrases from Mycobacterium tuberculosis with diazenylbenzenesulfonamides.EBI
Universita Degli Studi Di Firenze
The coumarin-binding site in carbonic anhydrase accommodates structurally diverse inhibitors: the antiepileptic lacosamide as an example and lead molecule for novel classes of carbonic anhydrase inhibitors.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors. Characterization and inhibition studies of the most active beta-carbonic anhydrase from Mycobacterium tuberculosis, Rv3588c.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors. Inhibition of the beta-class enzyme from the pathogenic yeast Candida glabrata with anions.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors. Inhibition of cytosolic isoforms I, II, III, VII and XIII with less investigated inorganic anions.EBI
Universita Degli Studi Di Firenze
A thiabendazole sulfonamide shows potent inhibitory activity against mammalian and nematode alpha-carbonic anhydrases.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors: design of spin-labeled sulfonamides incorporating TEMPO moieties as probes for cytosolic or transmembrane isozymes.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors: Inhibition of the new membrane-associated isoform XV with phenols.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrases as targets for medicinal chemistry.EBI
Universita Degli Studi Di Firenze
Phosph(on)ate as a zinc-binding group in metalloenzyme inhibitors: X-ray crystal structure of the antiviral drug foscarnet complexed to human carbonic anhydrase I.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors: inhibition of the cytosolic human isozyme VII with anions.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors: inhibition of the human isozymes I, II, VA, and IX with a library of substituted difluoromethanesulfonamides.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, IX, and XII with N-hydroxysulfamides--a new zinc-binding function in the design of inhibitors.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors. Inhibition of the human cytosolic isozyme VII with aromatic and heterocyclic sulfonamides.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors. Inhibition of the transmembrane isozyme XII with sulfonamides-a new target for the design of antitumor and antiglaucoma drugs?EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors. Inhibition of the membrane-bound human and bovine isozymes IV with sulfonamides.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with bis-sulfamates.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors. Inhibition of isozymes I, II, IV, V, and IX with anions isosteric and isoelectronic with sulfate, nitrate, and carbonate.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors: novel sulfonamides incorporating 1,3,5-triazine moieties as inhibitors of the cytosolic and tumour-associated carbonic anhydrase isozymes I, II and IX.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides derived from 4-isothiocyanato-benzolamide.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors: inhibition of the membrane-bound human isozyme IV with anions.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors. Inhibition of the newly isolated murine isozyme XIII with anions.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides incorporating 1,2,4-triazine moieties.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors. Inhibition of the beta-class enzyme from the methanoarchaeon Methanobacterium thermoautotrophicum (Cab) with anions.EBI
Universita Degli Studi Di Firenze
1,2,4-triazolo[4,3-a]quinoxalin-1-one moiety as an attractive scaffold to develop new potent and selective human A3 adenosine receptor antagonists: synthesis, pharmacological, and ligand-receptor modeling studies.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors: synthesis and topical intraocular pressure lowering effects of fluorine-containing inhibitors devoid of enhanced reactivity.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors. A general approach for the preparation of water-soluble sulfonamides incorporating polyamino-polycarboxylate tails and of their metal complexes possessing long-lasting, topical intraocular pressure-lowering properties.EBI
Universita Degli Studi Di Firenze
Nonaromatic sulfonamide group as an ideal anchor for potent human carbonic anhydrase inhibitors: role of hydrogen-bonding networks in ligand binding and drug design.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors: water-soluble 4-sulfamoylphenylthioureas as topical intraocular pressure-lowering agents with long-lasting effects.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors: perfluoroalkyl/aryl-substituted derivatives of aromatic/heterocyclic sulfonamides as topical intraocular pressure-lowering agents with prolonged duration of action.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors: inhibition of the tumor-associated isozyme IX with fluorine-containing sulfonamides. The first subnanomolar CA IX inhibitor discovered.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors: X-ray crystallographic structure of the adduct of human isozyme II with EMATE, a dual inhibitor of carbonic anhydrases and steroid sulfatase.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors: E7070, a sulfonamide anticancer agent, potently inhibits cytosolic isozymes I and II, and transmembrane, tumor-associated isozyme IX.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors: inhibition of the tumor-associated isozyme IX with aromatic and heterocyclic sulfonamides.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors: SAR and X-ray crystallographic study for the interaction of sugar sulfamates/sulfamides with isozymes I, II and IV.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors: inhibition of cytosolic isozymes I and II with sulfamide derivatives.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors. Preparation of potent sulfonamides inhibitors incorporating bile acid tails.EBI
Universita Degli Studi Di Firenze
Novel coumarins and 2-thioxo-coumarins as inhibitors of the tumor-associated carbonic anhydrases IX and XII.EBI
Universita Degli Studi Di Firenze
New chemotypes acting as isozyme-selective carbonic anhydrase inhibitors with low affinity for the offtarget cytosolic isoform II.EBI
Universita Degli Studi Di Firenze
5- and 6-membered (thio)lactones are prodrug type carbonic anhydrase inhibitors.EBI
Universita Degli Studi Di Firenze
Sulfonamides incorporating 1,3,5-triazine moieties selectively and potently inhibit carbonic anhydrase transmembrane isoforms IX, XII and XIV over cytosolic isoforms I and II: Solution and X-ray crystallographic studies.EBI
Universita Degli Studi Di Firenze
Design, synthesis and evaluation of N-benzoylindazole derivatives and analogues as inhibitors of human neutrophil elastase.EBI
Universita Degli Studi Di Firenze
Inhibition studies with anions and small molecules of two novel β-carbonic anhydrases from the bacterial pathogen Salmonella enterica serovar Typhimurium.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors. Inhibition of the β-class enzymes from the fungal pathogens Candida albicans and Cryptococcus neoformans with branched aliphatic/aromatic carboxylates and their derivatives.EBI
Universita Degli Studi Di Firenze
Purification and inhibition studies with anions and sulfonamides of ana-carbonic anhydrase from the Antarctic seal Leptonychotes weddellii.EBI
Universita Degli Studi Di Firenze
(R)-/(S)-10-camphorsulfonyl-substituted aromatic/heterocyclic sulfonamides selectively inhibit mitochondrial over cytosolic carbonic anhydrases.EBI
Universita Degli Studi Di Firenze
Inhibition ofß-carbonic anhydrases with ureido-substituted benzenesulfonamides.EBI
Universita Degli Studi Di Firenze
Polyamines inhibit carbonic anhydrases by anchoring to the zinc-coordinated water molecule.EBI
Universita Degli Studi Di Firenze
Inhibition studies of a beta-carbonic anhydrase from Brucella suis with a series of water soluble glycosyl sulfanilamides.EBI
Universita Degli Studi Di Firenze
The proteoglycan region of the tumor-associated carbonic anhydrase isoform IX acts as anintrinsic buffer optimizing CO2 hydration at acidic pH values characteristic of solid tumors.EBI
Universita Degli Studi Di Firenze
6-methyl-2,4-disubstituted pyridazin-3(2H)-ones: a novel class of small-molecule agonists for formyl peptide receptors.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors. Inhibition of the fungal beta-carbonic anhydrases from Candida albicans and Cryptococcus neoformans with boronic acids.EBI
Universita Degli Studi Di Firenze
Investigations of the esterase, phosphatase, and sulfatase activities of the cytosolic mammalian carbonic anhydrase isoforms I, II, and XIII with 4-nitrophenyl esters as substrates.EBI
Universita Degli Studi Di Firenze
Carbonic anhydrase inhibitors: the very weak inhibitors dithiothreitol, beta-mercaptoethanol, tris(carboxyethyl)phosphine and threitol interfere with the binding of sulfonamides to isozymes II and IX.EBI
Universita Degli Studi Di Firenze
3-hydroxy-quinazoline-2,4-dione as a useful scaffold to obtain selective Gly/NMDA and AMPA receptor antagonists.EBI
Universita Degli Studi Di Firenze
Synthesis and biological evaluation of analogues of 7-chloro-4,5-dihydro-4- oxo-8-(1,2,4-triazol-4-yl)-1,2,4-triazolo[1,5-a]quinoxaline-2-carboxylic acid (TQX-173) as novel selective AMPA receptor antagonists.EBI
Universita Degli Studi Di Firenze
Discovery of first-in-class multi-target adenosine AEBI
Universita Degli Studi Di Firenze
New 8-amino-1,2,4-triazolo[4,3-a]pyrazin-3-one derivatives. Evaluation of different moieties on the 6-aryl ring to obtain potent and selective human AEBI
Universita Degli Studi Di Firenze
Structural investigation on thiazolo[5,4-d]pyrimidines to obtain dual-acting blockers of CD73 and adenosine AEBI
Universita Degli Studi Di Firenze
Azidothymidine "Clicked" into 1,2,3-Triazoles: First Report on Carbonic Anhydrase-Telomerase Dual-Hybrid Inhibitors.EBI
Universita Degli Studi Di Firenze
Monothiocarbamates Strongly Inhibit Carbonic Anhydrases in Vitro and Possess Intraocular Pressure Lowering Activity in an Animal Model of Glaucoma.EBI
Universita Degli Studi Di Firenze
Modifications on the Amino-3,5-dicyanopyridine Core To Obtain Multifaceted Adenosine Receptor Ligands with Antineuropathic Activity.EBI
Universita Degli Studi Di Firenze
Synthesis and Evaluation of Carbonic Anhydrase Inhibitors with Carbon Monoxide Releasing Properties for the Management of Rheumatoid Arthritis.EBI
Universita Degli Studi Di Firenze
Novel human adenosine receptor antagonists based on the 7-amino-thiazolo[5,4-d]pyrimidine scaffold. Structural investigations at the 2-, 5- and 7-positions to enhance affinity and tune selectivity.EBI
Universita Degli Studi Di Firenze
Antioxidant-Conjugated 1,2,4-Triazolo[4,3-EBI
Universita Degli Studi Di Firenze
Fluorescent sulfonamide carbonic anhydrase inhibitors incorporating 1,2,3-triazole moieties: Kinetic and X-ray crystallographic studies.EBI
Universita Degli Studi Di Firenze
Anion and sulfonamide inhibition studies of an α-carbonic anhydrase from the Antarctic hemoglobinless fish Chionodraco hamatus.EBI
Universita Degli Studi Di Firenze
Combining the tail and the ring approaches for obtaining potent and isoform-selective carbonic anhydrase inhibitors: solution and X-ray crystallographic studies.EBI
Universita Degli Studi Di Firenze
Inhibition of human carbonic anhydrase isoforms I-XIV with sulfonamides incorporating fluorine and 1,3,5-triazine moieties.EBI
Universita Degli Studi Di Firenze
Structural study of the location of the phenyl tail of benzene sulfonamides and the effect on human carbonic anhydrase inhibition.EBI
Universita Degli Studi Di Firenze
7-Substituted-sulfocoumarins are isoform-selective, potent carbonic anhydrase II inhibitors.EBI
Universita Degli Studi Di Firenze
Functionalized pyrazoles and pyrazolo[3,4-d]pyridazinones: Synthesis and evaluation of their phosphodiesterase 4 inhibitory activity.EBI
Universita Degli Studi Di Firenze
4-Hydroxy-3-nitro-5-ureido-benzenesulfonamides Selectively Target the Tumor-Associated Carbonic Anhydrase Isoforms IX and XII Showing Hypoxia-Enhanced Antiproliferative Profiles.EBI
Universita Degli Studi Di Firenze
A new class of pyrazolo[5,1-c][1,2,4]triazines as γ-aminobutyric type A (GABAEBI
Universita Degli Studi Di Firenze
The aminopyridine-3,5-dicarbonitrile core for the design of new non-nucleoside-like agonists of the human adenosine AEBI
Universita Degli Studi Di Firenze
Structure-activity relationship studies and pharmacological characterization of NEBI
Universita Degli Studi Di Firenze
Design, synthesis and X-ray crystallography of selenides bearing benzenesulfonamide moiety with neuropathic pain modulating effects.EBI
Universita Degli Studi Di Firenze
Structural investigations on coumarins leading to chromeno[4,3-c]pyrazol-4-ones and pyrano[4,3-c]pyrazol-4-ones: New scaffolds for the design of the tumor-associated carbonic anhydrase isoforms IX and XII.EBI
Universita Degli Studi Di Firenze
Identification of novel thiazolo[5,4-d]pyrimidine derivatives as human AEBI
Universita Degli Studi Di Firenze
Development of novel pyridazinone-based adenosine receptor ligands.EBI
Universita Degli Studi Di Firenze
Synthesis and carbonic anhydrase inhibition of polycyclic imides incorporating N-benzenesulfonamide moieties.EBI
Universita Degli Studi Di Firenze
1,3-Oxazole-based selective picomolar inhibitors of cytosolic human carbonic anhydrase II alleviate ocular hypertension in rabbits: Potency is supported by X-ray crystallography of two leads.EBI
Universita Degli Studi Di Firenze
Bortezomib inhibits mammalian carbonic anhydrases.EBI
Universita Degli Studi Di Firenze
Imidazo[1,2-a]pyrazin-8-amine core for the design of new adenosine receptor antagonists: Structural exploration to target the AEBI
Universita Degli Studi Di Firenze
Synthesis of novel acyl selenoureido benzensulfonamides as carbonic anhydrase I, II, VII and IX inhibitors.EBI
Universita Degli Studi Di Firenze
Evaluation of selenide, diselenide and selenoheterocycle derivatives as carbonic anhydrase I, II, IV, VII and IX inhibitors.EBI
Universita Degli Studi Di Firenze
Synthesis of new 3-(2-mercapto-4-oxo-4H-quinazolin-3-yl)-benzenesulfonamides with strong inhibition properties against the tumor associated carbonic anhydrases IX and XII.EBI
Universita Degli Studi Di Firenze
Synthesis and carbonic anhydrase inhibition of a series of SLC-0111 analogs.EBI
Universita Degli Studi Di Firenze
N-substituted-5-substituted phthalamic acids as sortilin inhibitorsBDB
H. Lundbeck
Substituted 2-azabicycles and their use as orexin receptor modulatorsBDB
Janssen Pharmaceutica
Pyridine compounds and the uses thereofBDB
Purdue Pharma
Histone demethylase inhibitorsBDB
Celgene Quanticel Research
Compositions, synthesis, and methods of using phenylcycloalkylmethylamine derivativesBDB
Revivia Pharmaceuticals
Compounds having TRPV1 antagonistic activity and uses thereofBDB
Shionogi
Discovery of a selective inhibitor of oncogenic B-Raf kinase with potent antimelanoma activity.BDB
Plexxikon
Crystal structure of pyridoxal kinase in complex with roscovitine and derivatives.BDB
Chinese Academy of Sciences
Synthesis and antiviral activity of 4-benzyl pyridinone derivatives as potent and selective non-nucleoside human immunodeficiency virus type 1 reverse transcriptase inhibitors.BDB
Institut Curie
Pyrido[2,3-d]pyrimidin-7-one inhibitors of cyclin-dependent kinases.BDB
Parke-Davis Pharmaceutical Research
Tyrosine kinase inhibitors. 13. Structure-activity relationships for soluble 7-substituted 4-[(3-bromophenyl)amino]pyrido[4,3-d]pyrimidines designed as inhibitors of the tyrosine kinase activity of the epidermal growth factor receptor.BDB
University of Auckland
Tyrosine kinase inhibitors. 9. Synthesis and evaluation of fused tricyclic quinazoline analogues as ATP site inhibitors of the tyrosine kinase activity of the epidermal growth factor receptor.BDB
University of Auckland