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18 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Discovery of a new binding site on human choline kinasea1: design, synthesis, crystallographic studies, and biological evaluation of asymmetrical bispyridinium derivatives.EBI
Universidad De Granada
Scorpiand-like azamacrocycles prevent the chronic establishment of Trypanosoma cruzi in a murine model.EBI
Universidad De Granada
In vitro activity of scorpiand-like azamacrocycle derivatives in promastigotes and intracellular amastigotes of Leishmania infantum and Leishmania braziliensis.EBI
Universidad De Granada
Phthalazine derivatives containing imidazole rings behave as Fe-SOD inhibitors and show remarkable anti-T. cruzi activity in immunodeficient-mouse mode of infection.EBI
Universidad De Granada
In vitro and in vivo trypanosomicidal activity of pyrazole-containing macrocyclic and macrobicyclic polyamines: their action on acute and chronic phases of Chagas disease.EBI
Universidad De Granada
1,3,4-Thiadiazole derivatives as selective inhibitors of iNOS versus nNOS: Synthesis and structure-activity dependence.EBI
Universidad De Granada
Homodimeric bis-quaternary heterocyclic ammonium salts as potent acetyl- and butyrylcholinesterase inhibitors: a systematic investigation of the influence of linker and cationic heads over affinity and selectivity.EBI
Universidad De Granada
In vivo trypanosomicidal activity of imidazole- or pyrazole-based benzo[g]phthalazine derivatives against acute and chronic phases of Chagas disease.EBI
Universidad De Granada
New salicylic acid derivatives, double inhibitors of glycolate oxidase and lactate dehydrogenase, as effective agents decreasing oxalate production.EBI
Universidad De Granada
Symmetrical bis-quinolinium compounds: new human choline kinase inhibitors with antiproliferative activity against the HT-29 cell line.EBI
Universidad De Granada
Bispyridinium cyclophanes: novel templates for human choline kinase inhibitors.EBI
Universidad De Granada
Synthesis, bioevaluation and docking studies of new imidamide derivatives as nitric oxide synthase inhibitors.EBI
Universidad De Granada
Inhibition of nNOS activity in rat brain by synthetic kynurenines: structure-activity dependence.EBI
Universidad De Granada
-Alkyl Hydroxamates Display Potent and Selective Antileishmanial Activity.EBI
Universidad De Granada
Semi-synthesis of acylated triterpenes from olive-oil industry wastes for the development of anticancer and anti-HIV agents.EBI
Universidad De Granada
Synthesis and biological evaluation of 4,5-dihydro-1H-pyrazole derivatives as potential nNOS/iNOS selective inhibitors. Part 2: Influence of diverse substituents in both the phenyl moiety and the acyl group.EBI
Universidad De Granada
Salicylic Acid Derivatives Inhibit Oxalate Production in Mouse Hepatocytes with Primary Hyperoxaluria Type 1.EBI
Universidad De Granada
1,2-Diphenoxiethane salts as potent antiplasmodial agents.EBI
Universidad De Granada