PMID

Data

Article Title

Organization

Development of Glucose Regulated Protein 94-Selective Inhibitors Based on the BnIm and Radamide Scaffold.

The University of Kansas

Structure-Activity Relationships of the Peptide Kappa Opioid Receptor Antagonist Zyklophin.

The University of Kansas

Development of radamide analogs as Grp94 inhibitors.

The University of Kansas

Studies toward the Development of Antiproliferative Neoclerodanes from Salvinorin A.

The University of Kansas

Synthesis and¿-opioid receptor activity of furan-substituted salvinorin A analogues.

The University of Kansas

Are MDCK cells transfected with the human MRP2 gene a good model of the human intestinal mucosa?

The University of Kansas

Are MDCK cells transfected with the human MDR1 gene a good model of the human intestinal mucosa?

The University of Kansas

Semisynthetic neoclerodanes as kappa opioid receptor probes.

The University of Kansas

The sulfonimidamide as a novel transition state analog for aspartic acid and metallo proteases.

The University of Kansas

Identification and initial SAR of silybin: an Hsp90 inhibitor.

The University of Kansas

Discovery of dermorphin-based affinity labels with subnanomolar affinity for mu opioid receptors.

The University of Kansas

Design, synthesis, and pharmacological activities of dynorphin A analogues cyclized by ring-closing metathesis.

The University of Kansas

Synthesis of 4,5,6,7-tetrahydrothieno[3,2-c]pyridines and comparison with their isosteric 1,2,3,4-tetrahydroisoquinolines as inhibitors of phenylethanolamine N-methyltransferase.

The University of Kansas

Synthesis and pharmacological characterization of novel fluorescent histamine H2-receptor ligands derived from aminopotentidine.

The University of Kansas

High-throughput screening for Hsp90 ATPase inhibitors.

The University of Kansas

Conformational Constraint between Aromatic Residue Side Chains in the "Message" Sequence of the Peptide Arodyn Using Ring Closing Metathesis Results in a Potent and Selective Kappa Opioid Receptor Antagonist.

The University of Kansas

Fluoroalkylation of Dextromethorphan Improves CNS Exposure and Metabolic Stability.

The University of Kansas

Synthetic Studies of Neoclerodane Diterpenes from Salvia divinorum: Identification of a Potent and Centrally Acting μ Opioid Analgesic with Reduced Abuse Liability.

The University of Kansas

Design, synthesis, and biological evaluation of aminoalkylindole derivatives as cannabinoid receptor ligands with potential for treatment of alcohol abuse.

The University of Kansas

3D-QSAR Assisted Design, Synthesis and Evaluation of Novobiocin Analogues.

The University of Kansas

Isolation and characterization of Caco-2 subclones expressing high levels of multidrug resistance protein efflux transporter.

The University of Kansas

A functional assay for quantitation of the apparent affinities of ligands of P-glycoprotein in Caco-2 cells.

The University of Kansas

Click chemistry to probe Hsp90: Synthesis and evaluation of a series of triazole-containing novobiocin analogues.

The University of Kansas

Synthesis and evaluation of Hsp90 inhibitors that contain the 1,4-naphthoquinone scaffold.

The University of Kansas

Derrubone, an inhibitor of the Hsp90 protein folding machinery.

The University of Kansas

Resorcinol-Based Grp94-Selective Inhibitors.

The University of Kansas

Addressing Structural Flexibility at the A-Ring on Salvinorin A: Discovery of a Potent Kappa-Opioid Agonist with Enhanced Metabolic Stability.

The University of Kansas